SCHEMBL7200308

SCHEMBL7200308

CCc1c(C(=O)O)ccnc1-c1cc(C)c2nc(C)n(Cc3ncc(C(F)(F)F)cc3Cl)c2c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C19 P33261 1/20 0.37
MRGPRX4 Q96LA9 1/20 0.36
AGBL2 Q5U5Z8 1/20 0.36
GLA P06280 1/20 0.35
NPSR1 Q6W5P4 2/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
PIK3C2B O00750 2/20 0.34
EIF4EBP1 Q13541 1/20 0.33
KDM4E B2RXH2 2/20 0.33
ALDH1A1 P00352 2/20 0.33
ABCC3 O15438 1/20 0.33
ABCC4 O15439 1/20 0.33
USP2 O75604 1/20 0.33
ABCB11 O95342 1/20 0.33
CHRM2 P08172 1/20 0.33
ADRA2A P08913 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7195728 0.91 CYP1A2 (0.38) CYP3A4CYP1A2CYP2D6CYP2C19AGBL2
SCHEMBL7197594 0.85 MRGPRX4 (0.39) CYP3A4CYP1A2CYP2D6CYP2C19MRGPRX4
SCHEMBL6488962 0.84 MRGPRX4 (0.41) CYP3A4CYP1A2CYP2D6CYP2C19MRGPRX4
SCHEMBL7199966 0.83 CYP1A2 (0.38) CYP3A4CYP1A2CYP2D6CYP2C19AGBL2
SCHEMBL6490617 0.82 DCTPP1 (0.43) CYP3A4CYP1A2CYP2D6CYP2C19MRGPRX4
SCHEMBL7192311 0.82 CYP1A2 (0.38) CYP3A4CYP1A2CYP2D6CYP2C19MRGPRX4
SCHEMBL6502236 0.81 MRGPRX4 (0.39) CYP3A4CYP1A2CYP2D6CYP2C19MRGPRX4
SCHEMBL6488927 0.80 MRGPRX4 (0.44) CYP3A4CYP1A2CYP2D6CYP2C19MRGPRX4
SCHEMBL6490408 0.80 JMJD6 (0.41) CYP3A4CYP1A2CYP2D6CYP2C19MEN1
SCHEMBL6489988 0.79 DCTPP1 (0.40) CYP3A4CYP1A2CYP2D6CYP2C19MRGPRX4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004108686-A2 BENZIMIDAZOLE COMPOUNDS HAVING HYPOGLYCEMIC ACTIVITY FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2004-12-16 WO disclosed