SCHEMBL7202793

SCHEMBL7202793

CCC(Oc1ccc(NC(=O)NC(=O)c2cnc3c(c2)c(C)nn3C)cc1C(F)(F)F)C(=O)O

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 3/20 0.69
CCR5 P51681 3/20 0.69
S1PR1 P21453 5/20 0.40
SPR P35270 4/20 0.37
NR3C1 P04150 3/20 0.37
POLB P06746 1/20 0.36
BRAF P15056 2/20 0.36
ADRB2 P07550 1/20 0.36
GPR183 P32249 1/20 0.36
APLNR P35414 1/20 0.36
S1PR5 Q9H228 1/20 0.36
PDE5A O76074 1/20 0.35
KDR P35968 2/20 0.35
ABL1 P00519 1/20 0.35
LCK P06239 1/20 0.35
CSF1R P07333 1/20 0.35
LYN P07948 1/20 0.35
KIT P10721 1/20 0.35
SRC P12931 1/20 0.35
FLT1 P17948 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5961585 0.86 CCR2 (0.74) CCR2CCR5S1PR1SPRNR3C1
SCHEMBL5961562 0.84 CCR2 (0.71) CCR2CCR5S1PR1SPRNR3C1
SCHEMBL7163174 0.83 CCR2 (0.72) CCR2CCR5S1PR1SPRNR3C1
SCHEMBL18841095 0.82 CCR2 (1.00) CCR2CCR5SPRNR3C1POLB
SCHEMBL2863993 0.78 CCR2 (0.60) CCR2CCR5S1PR1NR3C1BRAF
SCHEMBL5961584 0.76 CCR2 (0.59) CCR2CCR5SPRNR3C1POLB
SCHEMBL5961499 0.76 CCR2 (0.59) CCR2CCR5SPRNR3C1POLB
SCHEMBL7079541 0.75 CCR2 (0.68) CCR2CCR5SPRNR3C1POLB
SCHEMBL5961458 0.73 CCR2 (0.68) CCR2CCR5SPRNR3C1POLB
SCHEMBL7079323 0.73 CCR2 (0.66) CCR2CCR5SPRNR3C1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1358188-A2 ANTAGONISTS OF MCP-1 FUNCTION AND METHODS OF USE THEREOF TELIK, INC. (US) 2003-11-05 EP claimed
WO-2002060900-A2 ANTAGONISTS OF MCP-1 FUNCTION AND METHODS OF USE THEREOF TELIK, INC. (US) 2002-08-08 WO claimed