SCHEMBL7204662

SCHEMBL7204662

CCCOC(=O)O[C@]1(C(=O)O)[C@H](C)C[C@H]2[C@@H]3CCC4=CC(=O)C=C[C@]4(C)[C@H]3CC[C@@]21C

nearest known ligand 0.52

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
LMNA P02545 4/20 0.51
MAPT P10636 2/20 0.51
NR3C1 P04150 4/20 0.46
PGR P06401 3/20 0.46
NR1I2 O75469 2/20 0.46
HIF1A Q16665 2/20 0.46
CNR1 P21554 1/20 0.46
CYP19A1 P11511 9/20 0.46
CYP3A4 P08684 2/20 0.46
ABCC3 O15438 1/20 0.44
ABCB11 O95342 1/20 0.44
USP2 O75604 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8587966 0.88 LMNA (0.54) LMNAMAPTNR3C1PGRNR1I2
SCHEMBL5672145 0.84 LMNA (0.52) LMNAMAPTNR3C1PGRNR1I2
SCHEMBL7877720 0.84 LMNA (0.52) LMNAMAPTNR3C1PGRNR1I2
SCHEMBL18662883 0.81 LMNA (0.52) LMNAMAPTNR3C1PGRNR1I2
SCHEMBL7135801 0.80 LMNA (0.49) LMNAMAPTNR3C1PGRNR1I2
SCHEMBL7137249 0.79 LMNA (0.48) LMNAMAPTNR3C1PGRNR1I2
SCHEMBL4220943 0.79 LMNA (0.52) LMNAMAPTNR3C1PGRNR1I2
SCHEMBL4218774 0.79 LMNA (0.52) LMNAMAPTNR3C1PGRNR1I2
SCHEMBL7136967 0.79 LMNA (0.48) LMNAMAPTNR3C1PGRNR1I2
SCHEMBL30915294 0.79 LMNA (0.48) LMNAMAPTCYP19A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6610675-B1 Identifying nontoxic therapeutically inactive metabolite of drug which elicits particular therapeutic response, converting inactive metabolite into activated structurally related drug species which cleaves in vivo to inactive metabolite Bodor, Nicholas S. 2003-08-26 US disclosed