SCHEMBL7205058

SCHEMBL7205058

COCCOCCOc1cc2ncnc(C3C(=O)Nc4ccc(S(N)(=O)=O)cc43)c2cc1OC

nearest known ligand 0.42

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
KDR P35968 18/20 0.42
EGFR P00533 1/20 0.39
ENPP1 P22413 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7209534 0.99 KDR (0.42) KDREGFRENPP1
SCHEMBL7207079 0.97 KDR (0.44) KDREGFR
Hydrochloric Acid SCHEMBL7210078 0.97 KDR (0.43) KDREGFR
SCHEMBL7205080 0.88 KDR (0.44) KDREGFR
SCHEMBL8501793 0.88 KDR (0.44) KDREGFR
Hydrochloric Acid SCHEMBL8501905 0.88 KDR (0.43) KDREGFR
Hydrochloric Acid SCHEMBL7206426 0.88 KDR (0.43) KDREGFR
SCHEMBL7206414 0.86 KDR (0.46) KDR
Hydrochloric Acid SCHEMBL7211167 0.85 KDR (0.45) KDR
SCHEMBL7205577 0.84 KDR (0.46) KDREGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0912557-B1 OXINDOLE DERIVATIVES ASTRAZENECA AB (SE) 2003-07-09 EP claimed
US-6265411-B1 ANGIOGENESIS INHIBITOR ZENECA LIMITED (GB) 2001-07-24 US claimed
EP-0912557-A1 OXINDOLE DERIVATIVES ZENECA LIMITED (GB) 1999-05-06 EP claimed
WO-1997042187-A1 OXINDOLE DERIVATIVES ZENECA LIMITED (GB) 1997-11-13 WO claimed
EP-0912557-B1 OXINDOLE DERIVATIVES ASTRAZENECA AB (SE) 2003-07-09 EP disclosed
US-6265411-B1 ANGIOGENESIS INHIBITOR ZENECA LIMITED (GB) 2001-07-24 US disclosed
EP-0912557-A1 OXINDOLE DERIVATIVES ZENECA LIMITED (GB) 1999-05-06 EP disclosed
WO-1997042187-A1 OXINDOLE DERIVATIVES ZENECA LIMITED (GB) 1997-11-13 WO disclosed