SCHEMBL7206

SCHEMBL7206

Cc1noc(-c2ccc(Br)cc2)c1C(CCCNS(C)(=O)=O)c1ccccc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.37
LPAR1 Q92633 3/20 0.37
LPAR3 Q9UBY5 1/20 0.37
BRD4 O60885 2/20 0.35
BRD2 P25440 2/20 0.35
BRD3 Q15059 2/20 0.35
EDNRB P24530 4/20 0.35
EDNRA P25101 4/20 0.35
NPY2R P49146 1/20 0.35
ALDH1A1 P00352 1/20 0.35
CYP2C9 P11712 2/20 0.35
ABCC3 O15438 1/20 0.35
ABCC4 O15439 1/20 0.35
ABCB11 O95342 1/20 0.35
CYP2C8 P10632 1/20 0.35
ABCB4 P21439 1/20 0.35
ABCC2 Q92887 1/20 0.35
SLCO1B3 Q9NPD5 1/20 0.35
SLCO1B1 Q9Y6L6 1/20 0.35
GAA P10253 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1379 0.82 GAA (0.39) LPAR1LPAR3BRD4NPY2RALDH1A1
SCHEMBL1464 0.79 GAA (0.38) LPAR1LPAR3EDNRBEDNRANPY2R
SCHEMBL1476 0.76 LPAR1 (0.43) LPAR1LPAR3BRD4ALDH1A1CYP2C9
SCHEMBL7205 0.76 BRD4 (0.40) POLBBRD4BRD2BRD3EDNRB
SCHEMBL4560 0.70 EDNRB (0.37) POLBEDNRBEDNRAALDH1A1CYP2C9
SCHEMBL4107 0.69 EDNRB (0.36) POLBBRD4EDNRBEDNRAALDH1A1
SCHEMBL6838 0.69 L3MBTL1 (0.40) LPAR1LPAR3BRD4BRD2BRD3
SCHEMBL1807 0.69 MEN1 (0.44) BRD4ALDH1A1LMNATDP1
SCHEMBL1166 0.68 LPAR1 (0.47) LPAR1LPAR3EDNRBEDNRAALDH1A1
SCHEMBL7770 0.68 ALDH1A1 (0.53) POLBLPAR1LPAR3ALDH1A1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2483252-A2 COMPOUNDS AS LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS Amira Pharmaceuticals, Inc. (US) 2012-08-08 EP disclosed
WO-2011041694-A2 COMPOUNDS AS LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS AMIRA PHARMACEUTICALS, INC. (US) 2011-04-07 WO disclosed