SCHEMBL7206020

SCHEMBL7206020

O=C(O)C[C@@H](NC(=O)CNC(=O)NCCCNc1nc2ccccc2[nH]1)c1ccc(-c2ccccc2)cc1

nearest known ligand 0.51

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 14/20 0.51
ITGAV P06756 14/20 0.51
ITGA2B P08514 3/20 0.51
ITGB5 P18084 3/20 0.51
ITGB6 P18564 2/20 0.51
KCNH2 Q12809 2/20 0.46
BCHE P06276 2/20 0.42
TRPC3 Q13507 1/20 0.42
TRPC4 Q9UBN4 1/20 0.42
TRPC5 Q9UL62 1/20 0.42
NPC1 O15118 1/20 0.41
HTT P42858 1/20 0.41
RAB9A P51151 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
CTSA P10619 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5845864 1.00 ITGB3 (0.51) ITGB3ITGAVITGA2BITGB5ITGB6
Trifluoroacetic Acid SCHEMBL5845761 0.95 ITGAV (0.47) ITGB3ITGAVITGA2BITGB5ITGB6
SCHEMBL5843698 0.95 ITGB3 (0.49) ITGB3ITGAVITGA2BITGB5ITGB6
Trifluoroacetic Acid SCHEMBL5844911 0.90 ITGAV (0.45) ITGB3ITGAVITGA2BITGB5ITGB6
SCHEMBL5845774 0.88 KCNH2 (0.43) ITGB3ITGAVITGA2BITGB5ITGB6
SCHEMBL6763140 0.85 ITGAV (0.56) ITGB3ITGAVITGA2BITGB5ITGB6
SCHEMBL5844227 0.85 ITGB3 (0.47) ITGB3ITGAVITGA2BITGB5ITGB6
SCHEMBL6762908 0.84 ITGAV (0.54) ITGB3ITGAVITGA2BITGB5ITGB6
SCHEMBL5844920 0.83 BCHE (0.44) ITGB3ITGAVITGA2BITGB5ITGB6
Trifluoroacetic Acid SCHEMBL6767494 0.81 ITGAV (0.52) ITGB3ITGAVITGA2BITGB5ITGB6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1343764-A1 UREA AND URETHANE DERIVATIVES AS INTEGRIN INHIBITORS MERCK PATENT GmbH (DE) 2003-09-17 EP claimed
WO-2002050039-A1 UREA AND URETHANE DERIVATIVES AS INTEGRIN INHIBITORS MERCK PATENT GMBH (DE) 2002-06-27 WO claimed
EP-1343764-A1 UREA AND URETHANE DERIVATIVES AS INTEGRIN INHIBITORS MERCK PATENT GmbH (DE) 2003-09-17 EP disclosed
WO-2002050039-A1 UREA AND URETHANE DERIVATIVES AS INTEGRIN INHIBITORS MERCK PATENT GMBH (DE) 2002-06-27 WO disclosed