SCHEMBL5845774

SCHEMBL5845774

O=C(CNC(=O)NCCCNc1nc2ccccc2[nH]1)NC(CC(=O)OC(=O)C(F)(F)F)c1ccc(-c2ccccc2)cc1

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.43
ITGAV P06756 13/20 0.41
ITGB3 P05106 12/20 0.41
ITGB6 P18564 3/20 0.41
ITGA2B P08514 2/20 0.41
ITGB5 P18084 2/20 0.41
BCHE P06276 2/20 0.39
ITGA5 P08648 3/20 0.37
ITGB1 P05556 2/20 0.37
ITGB8 P26012 1/20 0.37
TRPC3 Q13507 1/20 0.37
TRPC4 Q9UBN4 1/20 0.37
TRPC5 Q9UL62 1/20 0.37
NPC1 O15118 1/20 0.36
HTT P42858 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5844920 0.95 BCHE (0.44) KCNH2ITGAVITGB3ITGB6ITGA2B
Trifluoroacetic Acid SCHEMBL5845761 0.90 ITGAV (0.47) KCNH2ITGAVITGB3ITGB6ITGA2B
SCHEMBL5845534 0.89 BCHE (0.40) KCNH2ITGAVITGB3ITGB6ITGA2B
SCHEMBL7206020 0.88 ITGB3 (0.51) KCNH2ITGAVITGB3ITGB6ITGA2B
SCHEMBL5845864 0.88 ITGB3 (0.51) KCNH2ITGAVITGB3ITGB6ITGA2B
SCHEMBL6767502 0.87 ITGAV (0.42) KCNH2ITGAVITGB3ITGB6ITGA2B
SCHEMBL6763765 0.86 ITGAV (0.43) KCNH2ITGAVITGB3ITGB6ITGA2B
Trifluoroacetic Acid SCHEMBL5844911 0.85 ITGAV (0.45) KCNH2ITGAVITGB3ITGB6ITGA2B
SCHEMBL6762454 0.84 ITGAV (0.41) KCNH2ITGAVITGB3ITGB6ITGA2B
SCHEMBL5843698 0.83 ITGB3 (0.49) KCNH2ITGAVITGB3ITGB6ITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7135587-B2 Urea and urethane derivatives as integrin inhibitors MERCK PATENT GMBH (DE) 2006-11-14 US disclosed
EP-1343764-B1 UREA AND URETHANE DERIVATIVES AS INTEGRIN INHIBITORS MERCK PATENT GMBH (DE) 2004-08-25 EP disclosed
US-20040063644-A1 Urea and urethane derivatives as integrin inhibitors MERCK PATENT GMBH (DE) 2004-04-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040063644-A1 Urea and urethane derivatives as integrin inhibitors ITGB1, ITGB2, ITGA1 KCNH2 2038/4885ITGAV 16/4885ITGB3 7/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.