SCHEMBL7207282

SCHEMBL7207282

O=C(NCCc1ccccc1)[C@H](Cc1ccccc1)NC(=O)[C@H]1O[C@@H]1C(=O)O

nearest known ligand 0.55

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.54
CAPN1 P07384 5/20 0.50
CAPN9 O14815 1/20 0.50
CTSB P07858 1/20 0.50
MAPK1 P28482 1/20 0.50
PSMB1 P20618 1/20 0.48
PSMB5 P28074 1/20 0.48
PSMB2 P49721 1/20 0.48
MMP2 P08253 1/20 0.46
F10 P00742 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
MMP8 P22894 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7762733 1.00 KMT2A (0.54) KMT2ACAPN1CAPN9CTSBMAPK1
SCHEMBL8348444 1.00 KMT2A (0.54) KMT2ACAPN1CAPN9CTSBMAPK1
SCHEMBL7207278 1.00 KMT2A (0.54) KMT2ACAPN1CAPN9CTSBMAPK1
SCHEMBL8343183 1.00 KMT2A (0.54) KMT2ACAPN1CAPN9CTSBMAPK1
SCHEMBL7762722 1.00 KMT2A (0.54) KMT2ACAPN1CAPN9CTSBMAPK1
SCHEMBL9089190 0.89 CAPN1 (0.49) KMT2ACAPN1CAPN9CTSBMAPK1
SCHEMBL7206727 0.89 L3MBTL1 (0.59) CAPN1CAPN9CTSBMAPK1MMP2
SCHEMBL7206720 0.89 L3MBTL1 (0.59) CAPN1CAPN9CTSBMAPK1MMP2
SCHEMBL8349149 0.89 L3MBTL1 (0.59) CAPN1CAPN9CTSBMAPK1MMP2
SCHEMBL7762727 0.88 FCER2 (0.56) CAPN1PSMB5MMP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0921122-B1 EPOXYSUCCINAMIDE DERIVATIVES OR SALTS THEREOF TAIHO PHARMACEUTICAL CO LTD (JP) 2003-05-21 EP disclosed
EP-0808839-B1 EPOXYSUCCINAMIDE DERIVATIVES OR SALTS THEREOF, AND DRUGS CONTAINING THE SAME TAIHO PHARMACEUTICAL CO LTD (JP) 2001-05-23 EP disclosed
US-6110967-A USEFUL AS AGENTS FOR PREVENTING AND TREATING METABOLIC OSTEOPATHY SUCH AS OSTEOPOROSIS, HYPERCALCEMIA AND BONE METASTASIS OF CANCER BECAUSE THEY SPECIFICALLY INHIBITS CATHEPSIN L AND ITS FAMILY ENZYMES TO INHIBIT BONE RESORPTION TAIHO PHARMACEUTICALS CO., LTD. (JP) 2000-08-29 US disclosed
EP-0921122-A1 NOVEL EPOXYSUCCINAMIDE DERIVATIVES OR SALTS THEREOF TAIHO PHARMACEUTICAL COMPANY, LIMITED (JP) 1999-06-09 EP disclosed
EP-0808839-A1 EPOXYSUCCINAMIDE DERIVATIVES OR SALTS THEREOF, AND DRUGS CONTAINING THE SAME TAIHO PHARMACEUTICAL CO., LTD. (JP) 1997-11-26 EP disclosed