SCHEMBL7207416

SCHEMBL7207416

CCOC(=O)C(C(=O)OCC)C(C)(C)c1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIN1 Q13526 2/20 0.49
MEN1 O00255 3/20 0.47
KMT2A Q03164 3/20 0.47
NPC1 O15118 1/20 0.47
POLB P06746 2/20 0.46
MMP8 P22894 3/20 0.45
TSHR P16473 2/20 0.44
TDP1 Q9NUW8 1/20 0.44
SMN1; SMN2 Q16637 2/20 0.43
MAPT P10636 1/20 0.43
HTT P42858 1/20 0.43
HSD17B10 Q99714 1/20 0.43
CYP2C19 P33261 1/20 0.43
HIF1A Q16665 1/20 0.43
ALDH1A1 P00352 2/20 0.42
CHRM2 P08172 1/20 0.42
CHRM4 P08173 1/20 0.42
CHRM5 P08912 1/20 0.42
CHRM1 P11229 1/20 0.42
CHRM3 P20309 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7212419 0.93 PIN1 (0.46) PIN1MEN1KMT2ANPC1POLB
SCHEMBL7528311 0.90 PIN1 (0.44) PIN1MEN1KMT2ANPC1POLB
SCHEMBL9369385 0.84 PIN1 (0.47) PIN1MEN1KMT2ANPC1POLB
SCHEMBL12264169 0.84 MEN1 (0.53) PIN1MEN1KMT2ANPC1POLB
SCHEMBL1903612 0.83 CYP3A4 (0.50) MEN1KMT2APOLBTSHRTDP1
SCHEMBL22458448 0.83 NPSR1 (0.48) MEN1KMT2APOLBTSHRSMN1; SMN2
SCHEMBL7212428 0.83 PIN1 (0.46) PIN1MEN1KMT2ANPC1POLB
SCHEMBL8253229 0.83 MAPT (0.44) MEN1KMT2ANPC1POLBTDP1
SCHEMBL7213724 0.81 KMT2A (0.50) MEN1KMT2ATSHRMAPTCYP2C19
SCHEMBL13221585 0.81 ALDH1A1 (0.46) MEN1KMT2ANPC1POLBTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1854128-A Copper-catalyzed formation of carbon-heteroatom and carbon-carbon bonds MASSACHUSETTS INST TECHNOLOGY (US) 2006-11-01 CN disclosed
CN-1266112-C Copper-catalyzed carbon-heteroatom and carbon-carbon bond formation MASSACHUSETTS INST TECHNOLOGY (US) 2006-07-26 CN disclosed
US-6613934-B1 Enzymatic partial hydrolysis of a diester of malonic acid DEGUSSA AG (DE) 2003-09-02 US disclosed
EP-0812819-B1 Enantiomer-enriched tertiary hydrocarbonrest-substituted malonic acid ester and the preparation DEGUSSA (DE) 2001-11-28 EP disclosed
US-5831119-A Process for the preparation of aminoacetic acids with a tertiary hydrocarbon radical in the α-position, or their nitriles HUELS AKTIENGESELLSCHAFT (DE) 1998-11-03 US disclosed
EP-0812819-A2 Enantiomer-enriched tertiary hydrocarbonrest-substituted malonic acid ester and the preparation HÜLS AKTIENGESELLSCHAFT (DE) 1997-12-17 EP disclosed
US-5190922-A Antiinflammatory ABBOTT LABORATORIES (US) 1993-03-02 US disclosed
US-5063208-A Cardiovascular disorders, vision defects ABBOTT LABORATORIES (US) 1991-11-05 US disclosed
EP-0410260-A2 Peptidyl aminodiol renin inhibitors ABBOTT LABORATORIES (US) 1991-01-30 EP disclosed