SCHEMBL7208720

SCHEMBL7208720

COC(=O)[C@H](CC(C)C)NC(=O)N1CCC(Cc2ccccc2)CC1

nearest known ligand 0.72

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 4/20 0.72
KMT2A Q03164 4/20 0.72
POLB P06746 4/20 0.66
GAA P10253 1/20 0.62
SMN1; SMN2 Q16637 1/20 0.55
FAAH O00519 2/20 0.55
CYP3A4 P08684 1/20 0.54
CYP2D6 P10635 1/20 0.54
CYP2C9 P11712 1/20 0.54
CYP2C19 P33261 1/20 0.54
GFER P55789 1/20 0.54
TACR2 P21452 2/20 0.52
KCNH2 Q12809 1/20 0.52
HRH3 Q9Y5N1 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7209036 0.97 MEN1 (0.69) MEN1KMT2APOLBGAASMN1; SMN2
SCHEMBL4729475 0.87 POLB (0.71) MEN1KMT2APOLBGAAFAAH
SCHEMBL4725802 0.83 POLB (0.61) MEN1KMT2APOLBFAAHTACR2
SCHEMBL18396386 0.78 PSMB5 (0.62) KMT2APOLBGAA
SCHEMBL3598801 0.77 SLC6A2 (0.49) MEN1KMT2AKCNH2
SCHEMBL7037594 0.76 CACNA1B (0.60) POLBGAA
SCHEMBL7037597 0.76 CACNA1B (0.60) POLBGAA
SCHEMBL7342473 0.76 CACNA1B (0.60) POLBGAA
SCHEMBL18395980 0.76 PSMB5 (0.64) POLBGAASMN1; SMN2
SCHEMBL7345585 0.76 CACNA1B (0.68) POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6617426-B1 Peptide analogs of given formula; useful in treating neurodegenerative, autoimmune, cognitive disorders, stroke and traumatic injury MERCK SHARP & DOHME CORP. 2003-09-09 US disclosed
EP-1194443-A1 CYSTEINYL PROTEASE INHIBITORS Merck & Co., Inc. (US) 2002-04-10 EP disclosed
WO-2000078794-A1 CYSTEINYL PROTEASE INHIBITORS MERCK & CO., INC. (US) 2000-12-28 WO disclosed