SCHEMBL7209562

SCHEMBL7209562

CCOC(=O)c1ccccc1OC(=O)CCCCC(=O)Oc1ccccc1C(=O)OCC

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.61
KMT2A Q03164 2/20 0.61
KDM4E B2RXH2 1/20 0.61
RECQL P46063 1/20 0.61
TSHR P16473 4/20 0.61
ALDH1A1 P00352 4/20 0.53
MAPT P10636 3/20 0.53
HSD17B10 Q99714 1/20 0.53
PKM P14618 1/20 0.47
L3MBTL1 Q9Y468 3/20 0.46
TDP1 Q9NUW8 2/20 0.46
POLM Q9NP87 1/20 0.46
POLK Q9UBT6 1/20 0.46
POLL Q9UGP5 1/20 0.46
POLH Q9Y253 1/20 0.46
CYP3A4 P08684 2/20 0.46
USP2 O75604 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP2C9 P11712 1/20 0.46
ALOX15 P16050 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7892385 0.98 MEN1 (0.60) MEN1KMT2AKDM4ERECQLTSHR
SCHEMBL8499422 0.97 MEN1 (0.61) MEN1KMT2AKDM4ERECQLTSHR
SCHEMBL5706016 0.94 KDM4E (0.63) MEN1KMT2AKDM4ERECQLTSHR
SCHEMBL8498851 0.94 TSHR (0.65) MEN1KMT2AKDM4ERECQLTSHR
SCHEMBL7351148 0.91 KDM4E (0.56) MEN1KMT2AKDM4ERECQLTSHR
SCHEMBL14723637 0.89 KDM4E (0.51) MEN1KMT2AKDM4ERECQLTSHR
SCHEMBL13425197 0.89 HDAC1 (0.54) MEN1KMT2AKDM4ERECQLTSHR
SCHEMBL8500487 0.89 KDM4E (0.53) MEN1KMT2AKDM4ERECQLTSHR
SCHEMBL7360282 0.89 KDM4E (0.57) MEN1KMT2AKDM4ERECQLTSHR
SCHEMBL8587612 0.87 TSHR (0.65) MEN1KMT2AKDM4ERECQLTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1114841-B1 PROCESS FOR PRODUCING POLYARYLATE TEIJIN LTD (JP) 2003-10-08 EP disclosed
US-6417291-B1 CONDENSATION POLYMERIZATION AND ESTERIFICATION OF AROMATIC DIOL AND ESTER-FORMING MONOMER; ENDCAPPING WITH SALICYLIC ACID ESTER DERIVATIVE TEIJIN LIMITED (JP) 2002-07-09 US disclosed
US-6410777-B1 HALOGEN-FREE TEIJIN LIMITED (JP) 2002-06-25 US disclosed
US-6300459-B1 TRANSESTERIFYING AROMATIC POLYCARBONATE AND ACTIVE-HYDROGEN COMPOUND UNDER REDUCED PRESSURE FOLLOWED BY REACTION WITH SPECIFIED SALICYLIC ESTER DERIVATIVE TEIJIN LIMITED (JP) 2001-10-09 US disclosed
EP-1114841-A1 PROCESS FOR PRODUCING POLYARYLATE TEIJIN LIMITED (JP) 2001-07-11 EP disclosed
EP-0982340-A1 PROCESS FOR PRODUCING AROMATIC POLYCARBONATE TEIJIN LIMITED (JP) 2000-03-01 EP disclosed
EP-0980861-A1 SALICYLIC ESTER DERIVATIVES AND PROCESS FOR PRODUCING THE SAME TEIJIN LIMITED (JP) 2000-02-23 EP disclosed
EP-0764673-B1 Process for the production of polycarbonate TEIJIN LTD (JP) 1999-11-17 EP disclosed
US-5696222-A MELT POLYCONDENSATION OF AN AROMATIC DIHYDROXY COMPOUND AND DIPHENYLCARBONATE, THEN ADDING A SPECIFIC CARBONATE OR CARBOCYCLIC ESTER TO FORM TERMINAL BLOCKED POLYCARBONATE TEIJIN LIMITED (JP) 1997-12-09 US disclosed
EP-0764673-A2 Process for the production of polycarbonate TEIJIN LIMITED (JP) 1997-03-26 EP disclosed