SCHEMBL7210403

SCHEMBL7210403

Cc1ccncc1-c1cccn1-c1ccc(S(C)(=O)=O)cc1

nearest known ligand 0.59

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 17/20 0.59
PTGS1 P23219 2/20 0.47
MELK Q14680 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7215905 0.89 PTGS2 (0.58) PTGS2PTGS1
SCHEMBL7210775 0.80 PTGS2 (0.64) PTGS2PTGS1
SCHEMBL7211917 0.80 PTGS2 (0.70) PTGS2PTGS1MELK
SCHEMBL7210647 0.79 PTGS2 (0.58) PTGS2PTGS1
SCHEMBL7215899 0.77 PTGS2 (0.52) PTGS2PTGS1
SCHEMBL7210395 0.77 PTGS2 (0.70) PTGS2PTGS1MELK
SCHEMBL7210735 0.75 PTGS2 (0.59) PTGS2PTGS1
SCHEMBL7211965 0.75 PTGS2 (0.63) PTGS2PTGS1
SCHEMBL7216523 0.74 PTGS2 (0.59) PTGS2PTGS1
SCHEMBL5593921 0.73 PTGS2 (1.00) PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1369415-A1 Substituted pyrrolyl compounds for the treatment of inflammation G.D. SEARLE & CO. (US) 2003-12-10 EP claimed
EP-1369415-A1 Substituted pyrrolyl compounds for the treatment of inflammation G.D. SEARLE & CO. (US) 2003-12-10 EP disclosed
US-5935990-A PYRROLYL DERIVATIVES HAVING AT POSITION 1 OR 5 A PHENYL SUBSTITUTED WITH METHYLSULFONYL OR AMINOSULFONYL; INHIBIT CYCLOOXYGENASE-2 FOR USE TREATMENT OF INFLAMMATION, AS AN ANALGESIC, OR AS AN ANTIPYRETIC G.D. SEARLE & CO. (US) 1999-08-10 US disclosed