SCHEMBL7210775

SCHEMBL7210775

CS(=O)(=O)c1ccc(-n2cccc2-c2cccnc2)cc1

nearest known ligand 0.64

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 16/20 0.64
ALDH1A1 P00352 1/20 0.51
CYP2A6 P11509 1/20 0.51
CYP2A13 Q16696 1/20 0.51
PTGS1 P23219 6/20 0.50
FLT3 P36888 1/20 0.47
ALOX5 P09917 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7211965 0.89 PTGS2 (0.63) PTGS2ALDH1A1CYP2A6CYP2A13PTGS1
SCHEMBL7210405 0.86 PTGS2 (0.63) PTGS2ALDH1A1CYP2A6CYP2A13PTGS1
SCHEMBL7211917 0.86 PTGS2 (0.70) PTGS2PTGS1ALOX5
SCHEMBL7210395 0.83 PTGS2 (0.70) PTGS2PTGS1ALOX5
SCHEMBL7216523 0.83 PTGS2 (0.59) PTGS2PTGS1ALOX5
SCHEMBL7210403 0.80 PTGS2 (0.59) PTGS2PTGS1
SCHEMBL5594035 0.78 PTGS2 (1.00) PTGS2PTGS1
SCHEMBL5311655 0.78 PTGS2 (0.76) PTGS2PTGS1ALOX5
SCHEMBL5312538 0.78 PTGS2 (0.76) PTGS2PTGS1ALOX5
SCHEMBL5312009 0.78 PTGS2 (0.76) PTGS2PTGS1ALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1369415-A1 Substituted pyrrolyl compounds for the treatment of inflammation G.D. SEARLE & CO. (US) 2003-12-10 EP claimed
EP-1369415-A1 Substituted pyrrolyl compounds for the treatment of inflammation G.D. SEARLE & CO. (US) 2003-12-10 EP disclosed
US-5935990-A PYRROLYL DERIVATIVES HAVING AT POSITION 1 OR 5 A PHENYL SUBSTITUTED WITH METHYLSULFONYL OR AMINOSULFONYL; INHIBIT CYCLOOXYGENASE-2 FOR USE TREATMENT OF INFLAMMATION, AS AN ANALGESIC, OR AS AN ANTIPYRETIC G.D. SEARLE & CO. (US) 1999-08-10 US disclosed