SCHEMBL7210762

SCHEMBL7210762

Cc1csc(-n2cccc2-c2ccc(S(C)(=O)=O)cc2)c1

nearest known ligand 0.53

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 15/20 0.53
PTGS1 P23219 3/20 0.39
KCNH2 Q12809 2/20 0.38
ALOX5 P09917 1/20 0.38
CYP2C9 P11712 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5315712 0.88 PTGS2 (0.52) PTGS2PTGS1KCNH2ALOX5CYP2C9
SCHEMBL7216716 0.77 PTGS2 (0.60) PTGS2PTGS1CYP2C9
SCHEMBL7210860 0.76 PTGS2 (0.53) PTGS2PTGS1ALOX5
SCHEMBL5312538 0.76 PTGS2 (0.76) PTGS2PTGS1ALOX5CYP2C9
SCHEMBL5311655 0.76 PTGS2 (0.76) PTGS2PTGS1ALOX5CYP2C9
SCHEMBL5965033 0.73 PTGS2 (0.67) PTGS2PTGS1ALOX5CYP2C9
SCHEMBL5312009 0.73 PTGS2 (0.76) PTGS2PTGS1ALOX5
SCHEMBL7216668 0.73 PTGS2 (0.59) PTGS2PTGS1KCNH2ALOX5CYP2C9
SCHEMBL7216658 0.73 PTGS2 (0.52) PTGS2PTGS1KCNH2ALOX5CYP2C9
SCHEMBL348164 0.72 CA2 (0.44) PTGS2PTGS1KCNH2ALOX5CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1369415-A1 Substituted pyrrolyl compounds for the treatment of inflammation G.D. SEARLE & CO. (US) 2003-12-10 EP disclosed
US-5935990-A PYRROLYL DERIVATIVES HAVING AT POSITION 1 OR 5 A PHENYL SUBSTITUTED WITH METHYLSULFONYL OR AMINOSULFONYL; INHIBIT CYCLOOXYGENASE-2 FOR USE TREATMENT OF INFLAMMATION, AS AN ANALGESIC, OR AS AN ANTIPYRETIC G.D. SEARLE & CO. (US) 1999-08-10 US disclosed