SCHEMBL7210876

SCHEMBL7210876

Cc1ccncc1-n1c(C)ccc1-c1ccc(S(C)(=O)=O)cc1

nearest known ligand 0.56

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 16/20 0.56
KDM4E B2RXH2 1/20 0.53
ALDH1A1 P00352 1/20 0.53
MAPT P10636 1/20 0.53
HPGD P15428 1/20 0.53
PTGS1 P23219 2/20 0.45
MELK Q14680 1/20 0.41
IDO1 P14902 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7216743 0.81 PTGS2 (0.74) PTGS2KDM4EALDH1A1MAPTHPGD
SCHEMBL7210861 0.79 PTGS2 (0.71) PTGS2KDM4EALDH1A1MAPTHPGD
SCHEMBL7215899 0.78 PTGS2 (0.52) PTGS2PTGS1IDO1
SCHEMBL7215439 0.77 PTGS2 (0.60) PTGS2KDM4EALDH1A1MAPTHPGD
SCHEMBL7216175 0.74 PTGS2 (0.59) PTGS2KDM4EALDH1A1MAPTHPGD
SCHEMBL7216892 0.74 PTGS2 (0.67) PTGS2KDM4EALDH1A1MAPTHPGD
SCHEMBL7216986 0.72 PTGS2 (0.64) PTGS2KDM4EALDH1A1MAPTHPGD
SCHEMBL7210911 0.72 PTGS2 (0.64) PTGS2KDM4EALDH1A1MAPTHPGD
SCHEMBL7212097 0.72 PTGS2 (1.00) PTGS2KDM4EALDH1A1MAPTHPGD
SCHEMBL3831175 0.72 PTGS2 (1.00) PTGS2KDM4EALDH1A1MAPTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1369415-A1 Substituted pyrrolyl compounds for the treatment of inflammation G.D. SEARLE & CO. (US) 2003-12-10 EP claimed
EP-0946507-A1 SUBSTITUTED PYRROLYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1999-10-06 EP claimed
WO-1998025896-A1 SUBSTITUTED PYRROLYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1998-06-18 WO claimed
EP-1369415-A1 Substituted pyrrolyl compounds for the treatment of inflammation G.D. SEARLE & CO. (US) 2003-12-10 EP disclosed
US-5935990-A PYRROLYL DERIVATIVES HAVING AT POSITION 1 OR 5 A PHENYL SUBSTITUTED WITH METHYLSULFONYL OR AMINOSULFONYL; INHIBIT CYCLOOXYGENASE-2 FOR USE TREATMENT OF INFLAMMATION, AS AN ANALGESIC, OR AS AN ANTIPYRETIC G.D. SEARLE & CO. (US) 1999-08-10 US disclosed