SCHEMBL7216175

SCHEMBL7216175

Cc1cccnc1-n1c(C)ccc1-c1ccc(S(C)(=O)=O)cc1

nearest known ligand 0.59

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 13/20 0.59
ALDH1A1 P00352 2/20 0.47
KDM4E B2RXH2 1/20 0.47
MAPT P10636 1/20 0.47
HPGD P15428 1/20 0.47
PTGS1 P23219 2/20 0.43
HSD11B1 P28845 1/20 0.41
MAOB P27338 1/20 0.41
MYC P01106 1/20 0.40
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7215439 0.83 PTGS2 (0.60) PTGS2ALDH1A1KDM4EMAPTHPGD
SCHEMBL7210911 0.80 PTGS2 (0.64) PTGS2ALDH1A1KDM4EMAPTHPGD
SCHEMBL7211979 0.79 PTGS2 (0.53) PTGS2PTGS1HSD11B1MAOB
SCHEMBL7210861 0.76 PTGS2 (0.71) PTGS2ALDH1A1KDM4EMAPTHPGD
SCHEMBL7216743 0.75 PTGS2 (0.74) PTGS2ALDH1A1KDM4EMAPTHPGD
SCHEMBL3831175 0.75 PTGS2 (1.00) PTGS2ALDH1A1KDM4EMAPTHPGD
SCHEMBL21225774 0.74 MYC (0.58) ALDH1A1KDM4EMAPTHSD11B1MYC
SCHEMBL7210876 0.74 PTGS2 (0.56) PTGS2ALDH1A1KDM4EMAPTHPGD
SCHEMBL7211888 0.74 PTGS2 (0.59) PTGS2ALDH1A1KDM4EMAPTHPGD
SCHEMBL6517559 0.72 PTGS2 (0.89) PTGS2ALDH1A1KDM4EMAPTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1369415-A1 Substituted pyrrolyl compounds for the treatment of inflammation G.D. SEARLE & CO. (US) 2003-12-10 EP claimed
EP-0946507-A1 SUBSTITUTED PYRROLYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1999-10-06 EP claimed
WO-1998025896-A1 SUBSTITUTED PYRROLYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1998-06-18 WO claimed
EP-1369415-A1 Substituted pyrrolyl compounds for the treatment of inflammation G.D. SEARLE & CO. (US) 2003-12-10 EP disclosed
US-5935990-A PYRROLYL DERIVATIVES HAVING AT POSITION 1 OR 5 A PHENYL SUBSTITUTED WITH METHYLSULFONYL OR AMINOSULFONYL; INHIBIT CYCLOOXYGENASE-2 FOR USE TREATMENT OF INFLAMMATION, AS AN ANALGESIC, OR AS AN ANTIPYRETIC G.D. SEARLE & CO. (US) 1999-08-10 US disclosed