SCHEMBL7211481

SCHEMBL7211481

NS(=O)(=O)c1ccc(-c2ccccc2)c(-c2ccccc2C(F)(F)F)c1

nearest known ligand 0.49

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 7/20 0.49
PTGS1 P23219 6/20 0.49
CA2 P00918 5/20 0.46
CA1 P00915 4/20 0.46
CA5A P35218 1/20 0.46
CA5B Q9Y2D0 1/20 0.46
CA12 O43570 3/20 0.45
CA9 Q16790 3/20 0.45
KIF11 P52732 2/20 0.44
PDPK1 O15530 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
LRRK2 Q5S007 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1068740 0.85 CA12 (0.50) PTGS2PTGS1CA2CA1CA5A
Hydrochloric Acid SCHEMBL16015050 0.84 CA12 (0.49) PTGS2PTGS1CA2CA1CA12
SCHEMBL1068744 0.82 PTGS1 (0.62) PTGS2PTGS1CA2CA1CA5A
SCHEMBL4733933 0.81 CA2 (0.61) PTGS2PTGS1CA2CA1CA5A
SCHEMBL1069772 0.81 CA2 (0.51) CA2CA1CA5ACA5BCA12
Hydrochloric Acid SCHEMBL16015053 0.80 PTGS1 (0.60) PTGS2PTGS1CA2CA1CA5A
SCHEMBL30434205 0.80 CA2 (0.64) PTGS2PTGS1CA2CA1CA5A
SCHEMBL6794823 0.78 CA1 (0.66) PTGS2PTGS1CA2CA1CA12
SCHEMBL2452806 0.77 CA1 (0.41) PTGS2PTGS1CA2CA1CA5A
SCHEMBL7211494 0.77 CA2 (0.53) PTGS2PTGS1CA2CA1CA5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6613804-B2 Treatment of hypertension, cardiovascular disease, pulmonary hypertension, erythropoietin-mediated vasoconstriction, endotoxin shock, pulmonary hypertension, anaphylactic shock and hemorrhagic shock ENCYSIVE PHARMACEUTICALS, INC. 2003-09-02 US disclosed