SCHEMBL7211892

SCHEMBL7211892

Cc1c(S(=O)(=O)C(F)(F)F)cc(-c2ccc(S(N)(=O)=O)cc2)n1-c1ccc(F)cc1

nearest known ligand 0.81

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 14/20 0.81
CHRNA7 P36544 6/20 0.60
PTGS1 P23219 5/20 0.56
CYP2D6 P10635 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7210593 0.89 PTGS2 (1.00) PTGS2PTGS1
SCHEMBL7216763 0.83 CHRNA7 (0.62) PTGS2CHRNA7PTGS1
SCHEMBL7216536 0.82 PTGS2 (0.81) PTGS2CHRNA7PTGS1
SCHEMBL7216230 0.81 PTGS2 (0.79) PTGS2CHRNA7PTGS1CYP2D6
SCHEMBL7216281 0.80 PTGS2 (0.82) PTGS2CHRNA7CYP2D6
SCHEMBL7210628 0.79 CHRNA7 (0.62) PTGS2CHRNA7PTGS1
SCHEMBL7216202 0.76 PTGS2 (0.59) PTGS2CHRNA7PTGS1
SCHEMBL5311168 0.76 CHRNA7 (0.58) PTGS2CHRNA7PTGS1CYP2D6
SCHEMBL7210689 0.75 PTGS2 (0.77) PTGS2CHRNA7PTGS1
SCHEMBL3021555 0.75 PTGS2 (0.77) PTGS2CHRNA7PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1369415-A1 Substituted pyrrolyl compounds for the treatment of inflammation G.D. SEARLE & CO. (US) 2003-12-10 EP disclosed
US-5935990-A PYRROLYL DERIVATIVES HAVING AT POSITION 1 OR 5 A PHENYL SUBSTITUTED WITH METHYLSULFONYL OR AMINOSULFONYL; INHIBIT CYCLOOXYGENASE-2 FOR USE TREATMENT OF INFLAMMATION, AS AN ANALGESIC, OR AS AN ANTIPYRETIC G.D. SEARLE & CO. (US) 1999-08-10 US disclosed