SCHEMBL7212062

SCHEMBL7212062

COc1ccc(S(=O)(=O)CC[C@H](C)O)cc1

nearest known ligand 0.71

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MMP13 P45452 8/20 0.71
MMP1 P03956 5/20 0.71
HTT P42858 1/20 0.59
NPSR1 Q6W5P4 1/20 0.59
MMP8 P22894 2/20 0.57
MEN1 O00255 2/20 0.52
KMT2A Q03164 2/20 0.52
PKM P14618 2/20 0.48
CA1 P00915 1/20 0.46
CA2 P00918 1/20 0.46
MMP2 P08253 1/20 0.46
MMP9 P14780 1/20 0.46
GAA P10253 1/20 0.46
POLB P06746 1/20 0.46
MAPT P10636 1/20 0.46
ALDH1A1 P00352 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7212058 1.00 MMP13 (0.71) MMP13MMP1HTTNPSR1MMP8
SCHEMBL8204581 1.00 MMP13 (0.71) MMP13MMP1HTTNPSR1MMP8
SCHEMBL29296550 0.86 MMP13 (0.76) MMP13MMP1HTTNPSR1MMP8
SCHEMBL7212305 0.83 MMP13 (1.00) MMP13MMP1HTTNPSR1MMP8
SCHEMBL8206303 0.83 MMP13 (1.00) MMP13MMP1HTTNPSR1MMP8
SCHEMBL8206300 0.83 MMP13 (1.00) MMP13MMP1HTTNPSR1MMP8
SCHEMBL7207704 0.83 MMP13 (0.66) MMP13MMP1HTTNPSR1MMP8
SCHEMBL7400878 0.83 MMP13 (0.66) MMP13MMP1HTTNPSR1MMP8
SCHEMBL7207701 0.83 MMP13 (0.66) MMP13MMP1HTTNPSR1MMP8
SCHEMBL7924711 0.83 MMP2 (0.63) MMP13MMP1HTTMMP8MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0939628-B1 THIOL SULFONE METALLOPROTEASE INHIBITORS MONSANTO CO (US) 2003-03-05 EP disclosed
US-6013649-A BOND DISORDERS; AUTOIMMUNE DISEASES; ANTITUMOR AGENTS MONSANTO COMPANY (US) 2000-01-11 US disclosed
EP-0939628-A4 THIOL SULFONE METALLOPROTEASE INHIBITORS MONSANTO CO (US) 1999-12-22 EP disclosed
EP-0939628-A1 THIOL SULFONE METALLOPROTEASE INHIBITORS MONSANTO COMPANY (US) 1999-09-08 EP disclosed
WO-1998003164-A1 THIOL SULFONE METALLOPROTEASE INHIBITORS MONSANTO COMPANY (US) 1998-01-29 WO disclosed