SCHEMBL7212183

SCHEMBL7212183

CCCN(CCC)C(=O)N(C)c1nc(-c2ccccc2)ncc1C(=O)O

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.53
SMN1; SMN2 Q16637 4/20 0.53
MEN1 O00255 7/20 0.47
KMT2A Q03164 7/20 0.47
MAPT P10636 2/20 0.44
LMNA P02545 1/20 0.44
MAPK1 P28482 1/20 0.44
ATM Q13315 1/20 0.44
HPGD P15428 2/20 0.44
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
TP53 P04637 1/20 0.44
FOS P01100 2/20 0.43
JUN P05412 2/20 0.43
NFKB1 P19838 2/20 0.43
NFKB2 Q00653 2/20 0.43
RELA Q04206 2/20 0.43
KDM4E B2RXH2 2/20 0.43
CYP1A2 P05177 1/20 0.41
POLB P06746 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27999147 0.85 ALDH1A1 (0.48) ALDH1A1SMN1; SMN2MEN1KMT2AMAPT
SCHEMBL7217021 0.81 ALDH1A1 (0.50) ALDH1A1SMN1; SMN2MEN1KMT2AMAPT
SCHEMBL8294634 0.79 ALDH1A1 (0.69) ALDH1A1SMN1; SMN2MEN1KMT2AMAPT
SCHEMBL7212190 0.74 SMN1; SMN2 (0.46) ALDH1A1SMN1; SMN2MEN1KMT2AMAPT
SCHEMBL12929899 0.73 ALDH1A1 (0.67) ALDH1A1SMN1; SMN2MEN1KMT2AMAPT
SCHEMBL12929356 0.73 ALDH1A1 (0.67) ALDH1A1SMN1; SMN2MEN1KMT2AMAPT
SCHEMBL7210402 0.71 ALDH1A1 (0.71) ALDH1A1SMN1; SMN2MEN1KMT2AMAPT
SCHEMBL8295375 0.70 ALDH1A1 (0.67) ALDH1A1SMN1; SMN2MEN1KMT2AMAPT
SCHEMBL8294606 0.69 MEN1 (0.60) ALDH1A1SMN1; SMN2MEN1KMT2ALMNA
SCHEMBL8294641 0.69 ALDH1A1 (1.00) ALDH1A1SMN1; SMN2MEN1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1036794-B1 2-ARYL-8-OXODIHYDROPURINE DERIVATIVES, PROCESS FOR PRODUCING THE SAME, MEDICINAL COMPOSITIONS CONTAINING THE SAME, AND INTERMEDIATES THEREOF DAINIPPON PHARMACEUTICAL CO (JP) 2003-08-27 EP disclosed
US-6372740-B1 NERVOUS SYSTEM DISORDERS, ANTIEPILEPTIC AGENTS AND ANTIDEPRESSANTS DAINIPPON PHARMACEUTICAL CO., LTD. (JP) 2002-04-16 US disclosed
EP-1036794-A1 2-ARYL-8-OXODIHYDROPURINE DERIVATIVES, PROCESS FOR PRODUCING THE SAME, MEDICINAL COMPOSITIONS CONTAINING THE SAME, AND INTERMEDIATES THEREOF Dainippon Pharmaceutical Co., Ltd. (JP) 2000-09-20 EP disclosed