SCHEMBL7212252

SCHEMBL7212252

O=C(NC1N=C(c2ccccc2F)c2ccccc2N(CC(F)(F)F)C1=O)c1ccc(Cl)c(Cl)c1

nearest known ligand 0.64

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CCKAR P32238 16/20 0.64
CCKBR P32239 16/20 0.64
KCNH2 Q12809 2/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8761262 0.88 CCKAR (0.64) CCKARCCKBR
SCHEMBL8846479 0.85 CCKBR (0.64) CCKARCCKBRKCNH2
SCHEMBL9533402 0.83 CCKAR (0.59) CCKARCCKBR
SCHEMBL8761256 0.82 CCKAR (0.62) CCKARCCKBR
SCHEMBL6005837 0.81 KCNH2 (0.53) CCKARCCKBRKCNH2
SCHEMBL8846319 0.79 KCNH2 (0.77) CCKARCCKBRKCNH2
SCHEMBL8462639 0.79 KCNH2 (0.77) CCKARCCKBRKCNH2
SCHEMBL9526892 0.78 CCKBR (1.00) CCKARCCKBR
SCHEMBL9526889 0.78 CCKBR (1.00) CCKARCCKBR
SCHEMBL8462710 0.77 KCNH2 (0.81) KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0907644-A4 PHARMACEUTICAL PREPARATION MERCK & CO INC (US) 2003-02-05 EP claimed
EP-0907644-A1 PHARMACEUTICAL PREPARATION Merck & Co., Inc. (US) 1999-04-14 EP claimed
WO-1998000405-A1 PHARMACEUTICAL PREPARATION MERCK & CO., INC. (US) 1998-01-08 WO claimed
EP-0776208-A4 2,3-DIHYDRO-1-(2,2,2-TRIFLUOROETHYL)-2-OXO-5-PHENYL-1H-1,4-BENZODIAZEPINES MERCK & CO INC (US) 1997-12-29 EP disclosed
US-5658901-A 2,3-dihydro-1-(2,2,2,-trifluoroethyl)-2-oxo-5-phenyl-1H-1,4-benzodiazepines MERCK & CO., INC. (US) 1997-08-19 US disclosed
EP-0776208-A1 2,3-DIHYDRO-1-(2,2,2-TRIFLUOROETHYL)-2-OXO-5-PHENYL-1H-1,4-BENZODIAZEPINES MERCK & CO. INC. (US) 1997-06-04 EP disclosed
WO-1996005839-A1 2,3-DIHYDRO-1-(2,2,2-TRIFLUOROETHYL)-2-OXO-5-PHENYL-1H-1,4-BENZODIAZEPINES MERCK & CO., INC. (US) 1996-02-29 WO disclosed