SCHEMBL7212287

SCHEMBL7212287

CC(=O)N(c1cccc(C(F)(F)F)c1C(F)(F)F)[C@H]1N=C(c2ccccc2)c2ccccc2N(CC(F)(F)F)C1=O

nearest known ligand 0.51

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 3/20 0.51
CALCRL Q16602 17/20 0.43
RAMP1 O60894 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3252895 0.72 KCNH2 (0.47) KCNH2CALCRLRAMP1
SCHEMBL7744132 0.72 KCNH2 (0.45) KCNH2
SCHEMBL7744591 0.72 KCNH2 (0.45) KCNH2
SCHEMBL3247608 0.72 KCNH2 (0.57) KCNH2CALCRLRAMP1
SCHEMBL8462992 0.72 KCNH2 (0.82) KCNH2CALCRLRAMP1
SCHEMBL3859605 0.70 GABRP (0.61) KCNH2CALCRLRAMP1
SCHEMBL1834474 0.70 GABRP (0.61) KCNH2CALCRLRAMP1
SCHEMBL8223082 0.68 KCNH2 (0.73) KCNH2CALCRLRAMP1
L-768673 SCHEMBL7207125 0.67 KCNH2 (1.00) KCNH2CALCRLRAMP1
SCHEMBL8462904 0.67 KCNH2 (0.77) KCNH2CALCRLRAMP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0907644-A4 PHARMACEUTICAL PREPARATION MERCK & CO INC (US) 2003-02-05 EP disclosed
EP-0907644-A1 PHARMACEUTICAL PREPARATION Merck & Co., Inc. (US) 1999-04-14 EP disclosed
WO-1998000405-A1 PHARMACEUTICAL PREPARATION MERCK & CO., INC. (US) 1998-01-08 WO disclosed