SCHEMBL7212295

SCHEMBL7212295

OC(c1ccccn1)c1cc(C(F)(F)F)nc2ccccc12

nearest known ligand 0.69

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 2/20 0.69
ADORA1 P30542 1/20 0.69
MAPT P10636 2/20 0.46
IGF1R P08069 4/20 0.42
TLR7 Q9NYK1 1/20 0.42
ADRB2 P07550 1/20 0.40
RECQL P46063 1/20 0.39
MAPK1 P28482 1/20 0.39
TACR3 P29371 1/20 0.37
GAA P10253 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
KMT2A Q03164 2/20 0.36
CYP1A2 P05177 2/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
BLM P54132 1/20 0.36
BACE1 P56817 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7288128 0.83 KCNH2 (0.52) ADORA2AADORA1MAPTGAACYP1A2
SCHEMBL8941191 0.83 KCNH2 (0.52) ADORA2AADORA1MAPTGAACYP1A2
SCHEMBL7278581 0.83 KCNH2 (0.52) ADORA2AADORA1MAPTGAACYP1A2
SCHEMBL7226777 0.82 ADORA2A (1.00) ADORA2AADORA1MAPTIGF1RTLR7
SCHEMBL7208784 0.80 MAPT (0.49) ADORA2AADORA1MAPTRECQLTACR3
SCHEMBL8441818 0.77 ADORA2A (0.71) ADORA2AADORA1MAPTIGF1RTLR7
SCHEMBL7225702 0.76 MAPT (0.46) ADORA2AADORA1MAPTRECQLTACR3
SCHEMBL19150082 0.75 ADORA2A (0.68) ADORA2AADORA1MAPTIGF1RTLR7
SCHEMBL14424722 0.75 MAPT (0.56) MAPTRECQLNPSR1KMT2ACYP1A2
SCHEMBL14424717 0.75 MAPT (0.56) MAPTRECQLNPSR1KMT2ACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6608085-B1 Administering for neuroprotection VERNALIS RESEARCH LIMITED (GB) 2003-08-19 US disclosed
EP-1107761-A2 4-QUINOLINEMETHANOL DERIVATIVES AS PURINE RECEPTOR ANTAGONISTS (II) VERNALIS RESEARCH LIMITED (GB) 2001-06-20 EP disclosed
WO-2000013682-A2 4-QUINOLINEMETHANOL DERIVATIVES AS PURINE RECEPTOR ANTAGONISTS.(II) VERNALIS RESEARCH LIMITED (GB) 2000-03-16 WO disclosed