SCHEMBL7225702

SCHEMBL7225702

COc1cc(C(O)c2ccccn2)c2ccccc2n1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.46
NPC1 O15118 1/20 0.41
TACR3 P29371 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
ADORA2A P29274 1/20 0.39
ADORA1 P30542 1/20 0.39
CYP3A4 P08684 1/20 0.39
PDE10A Q9Y233 1/20 0.39
AHR P35869 2/20 0.38
HTR3E A5X5Y0 1/20 0.38
HTR3B O95264 1/20 0.38
HTR3A P46098 1/20 0.38
HTR3D Q70Z44 1/20 0.38
HTR3C Q8WXA8 1/20 0.38
SCD O00767 1/20 0.37
LMNA P02545 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
POLB P06746 1/20 0.37
ACHE P22303 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7207260 0.83 CYP3A4 (0.45) MAPTMEN1KMT2ACYP3A4PDE10A
SCHEMBL7225962 0.82 ADORA2A (0.57) NPC1MEN1KMT2AADORA2AADORA1
SCHEMBL15212407 0.81 ACP1 (0.56) MAPTNPC1TACR3LMNAALDH1A1
SCHEMBL7208784 0.80 MAPT (0.49) MAPTTACR3ADORA2AADORA1RECQL
SCHEMBL7212295 0.76 ADORA2A (0.69) MAPTTACR3KMT2AADORA2AADORA1
SCHEMBL16307497 0.76 KDM4E (0.49) MAPTNPC1TACR3MEN1KMT2A
SCHEMBL16019540 0.75 BCL2L1 (0.47) MAPTNPC1MEN1KMT2AHTR3E
SCHEMBL14424722 0.75 MAPT (0.56) MAPTNPC1MEN1KMT2ACYP3A4
SCHEMBL14424717 0.75 MAPT (0.56) MAPTNPC1MEN1KMT2ACYP3A4
SCHEMBL7221180 0.74 ADORA2A (0.43) NPC1TACR3MEN1KMT2AADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6583156-B1 Particularly adenosine A2A receptors; neurodegenerative disorders; 2,8-bis(trifluoromethyl)-alpha -(3-thienyl)-4-quinolinemethanol VERNALIS RESEARCH LIMITED (GB) 2003-06-24 US disclosed