SCHEMBL7212912

SCHEMBL7212912

COc1ccc(-c2c[nH]c(N)c2)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 3/20 0.47
MAPK1 P28482 2/20 0.46
NPC1 O15118 1/20 0.46
TP53 P04637 1/20 0.46
CASP3 P42574 1/20 0.46
RAB9A P51151 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
SENP8 Q96LD8 1/20 0.46
SENP7 Q9BQF6 1/20 0.46
SENP6 Q9GZR1 1/20 0.46
ESR2 Q92731 1/20 0.45
TDP1 Q9NUW8 2/20 0.45
ALDH1A1 P00352 1/20 0.43
CYP3A4 P08684 1/20 0.43
MAOB P27338 2/20 0.43
ABL1 P00519 1/20 0.43
ABCB1 P08183 1/20 0.43
BCR P11274 1/20 0.43
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10999330 0.79 TTK (0.62) DYRK1AMAPK1NPC1TP53CASP3
SCHEMBL6152523 0.78 KDM4E (0.50) DYRK1AMAPK1NPC1TP53CASP3
SCHEMBL2214586 0.74
SCHEMBL197522 0.73 CA1 (0.79) DYRK1AMAPK1NPC1TP53CASP3
SCHEMBL6733562 0.73 CA1 (0.79) DYRK1AMAPK1NPC1TP53CASP3
SCHEMBL9151672 0.73 CA1 (0.79) DYRK1AMAPK1NPC1TP53CASP3
SCHEMBL28326433 0.73 ACHE (0.52) DYRK1AMAPK1NPC1TP53CASP3
SCHEMBL20392617 0.73 SCN2A (0.50) DYRK1ANPC1CASP3RAB9ASMN1; SMN2
SCHEMBL19664327 0.73 SCN2A (0.50) DYRK1ANPC1CASP3RAB9ASMN1; SMN2
SCHEMBL1926936 0.72 TDP1 (0.84) DYRK1AMAPK1NPC1TP53CASP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1283832-A1 INHIBITORS OF 11-BETA-HYDROXY STEROID DEHYDROGENASE TYPE 1 BIOVITRUM AB (SE) 2003-02-19 EP disclosed
WO-2001090092-A1 INHIBITORS OF 11-BETA-HYDROXY STEROID DEHYDROGENASE TYPE 1 BIOVITRUM AB (SE) 2001-11-29 WO disclosed