SCHEMBL7212985

SCHEMBL7212985

O=C(NO)C1(NS(=O)(=O)c2ccc(OCc3ccc(Cl)cc3F)cc2)COC(CCCO)C1

nearest known ligand 0.51

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MMP1 P03956 12/20 0.51
MMP13 P45452 11/20 0.51
ADAM17 P78536 5/20 0.47
ADAMTS7 Q9UKP4 1/20 0.46
ADAMTS5 Q9UNA0 1/20 0.46
ADAMTS4 O75173 3/20 0.44
MMP2 P08253 2/20 0.44
MMP3 P08254 1/20 0.44
MMP9 P14780 1/20 0.44
MMP12 P39900 1/20 0.44
MMP14 P50281 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7208099 0.92 MMP1 (0.52) MMP1MMP13ADAM17ADAMTS7ADAMTS5
SCHEMBL7214333 0.90 MMP1 (0.48) MMP1MMP13ADAM17ADAMTS7ADAMTS5
SCHEMBL7214298 0.87 MMP1 (0.49) MMP1MMP13ADAM17ADAMTS7ADAMTS5
SCHEMBL7212989 0.87 MMP1 (0.54) MMP1MMP13ADAM17ADAMTS7ADAMTS5
SCHEMBL7214292 0.84 MMP1 (0.49) MMP1MMP13ADAM17ADAMTS7ADAMTS5
SCHEMBL7209165 0.83 MMP1 (0.53) MMP1MMP13ADAM17ADAMTS7ADAMTS5
SCHEMBL7213082 0.82 MMP1 (0.53) MMP1MMP13ADAM17ADAMTS7ADAMTS5
SCHEMBL7214324 0.81 MMP1 (0.50) MMP1MMP13ADAM17ADAMTS7ADAMTS5
SCHEMBL7208565 0.81 MMP1 (0.49) MMP1MMP13ADAM17ADAMTS7ADAMTS5
SCHEMBL7510613 0.80 MMP1 (0.42) MMP1MMP13ADAM17ADAMTS7ADAMTS5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1181285-B1 3-(ARYLSULFONYLAMINO)-TETRAHYDROFURAN-3-CARBOXYLIC ACID HYDROXAMIDES PFIZER PROD INC (US) 2003-10-08 EP disclosed
EP-1181285-A2 3-(ARYLSULFONYLAMINO)-TETRAHYDROFURAN-3-CARBOXYLIC ACID HYDROXAMIDES Pfizer Products Inc. (US) 2002-02-27 EP disclosed
US-6342521-B1 DRUGS FOR TREATMENT OF ARTHRITIS PFIZER INC. 2002-01-29 US disclosed
WO-2000073294-A2 3-(ARYLSULFONYLAMINO)-TETRAHYDROFURAN-3-CARBOXYLIC ACID HYDROXAMIDES PFIZER PRODUCTS INC. (US) 2000-12-07 WO disclosed