SCHEMBL7213853

SCHEMBL7213853

COc1ccc(C(=O)NC(C)(C#N)C(C)C)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.50
CA1 P00915 3/20 0.49
CA2 P00918 3/20 0.49
PLK1 P53350 1/20 0.49
NPC1 O15118 4/20 0.46
RAB9A P51151 4/20 0.46
SMN1; SMN2 Q16637 3/20 0.46
ALOX15 P16050 2/20 0.46
TP53 P04637 2/20 0.46
L3MBTL1 Q9Y468 3/20 0.46
GAA P10253 2/20 0.46
KDM4E B2RXH2 1/20 0.46
HTT P42858 1/20 0.46
ALDH1A1 P00352 2/20 0.46
LMNA P02545 2/20 0.46
APEX1 P27695 1/20 0.46
MAPK1 P28482 1/20 0.46
RECQL P46063 1/20 0.46
HSD17B10 Q99714 1/20 0.46
TDP1 Q9NUW8 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7220101 0.84 HPGD (0.46) MAPTNPC1RAB9ASMN1; SMN2GAA
SCHEMBL7214349 0.82 POLB (0.47) MAPTNPC1RAB9ASMN1; SMN2L3MBTL1
SCHEMBL7213607 0.82 POLB (0.49) CA1SMN1; SMN2ALOX15KDM4EALDH1A1
SCHEMBL15526785 0.80 MAPT (0.57) MAPTCA1CA2PLK1NPC1
SCHEMBL7219751 0.80 HTT (0.54) MAPTNPC1SMN1; SMN2KDM4EHTT
SCHEMBL6418333 0.76 MAPT (0.64) MAPTCA1CA2PLK1NPC1
SCHEMBL8014083 0.75 MAPT (0.62) MAPTCA1CA2PLK1NPC1
SCHEMBL3286749 0.74 CYP2B6 (0.48) MAPTRAB9ASMN1; SMN2L3MBTL1HTT
SCHEMBL28456891 0.72 MAPT (0.58) MAPTCA1CA2PLK1NPC1
SCHEMBL11665996 0.72 CA1 (0.61) MAPTCA1CA2PLK1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6504046-B1 Cyclization of nitriles using acids, to form oxazolinone chemical intermediates such as 2-phenyl-4-isopropyl-4-methyl-1,3-oxazol-5-one, used as fungicides IHARA CHEMICAL INDUSTRY CO., LTD. (JP) 2003-01-07 US disclosed
EP-1092705-A1 PROCESS FOR THE PREPARATION OF AMIDES IHARA CHEMICAL INDUSTRY Co., Ltd. (JP) 2001-04-18 EP disclosed