SCHEMBL7214920

SCHEMBL7214920

CC(=O)N1CCc2c(C)ccnc21

nearest known ligand 0.54

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 12/20 0.54
CYP11B2 P19099 5/20 0.42
HTR2A P28223 1/20 0.42
HTR2C P28335 1/20 0.42
HTR2B P41595 1/20 0.42
CYP11B1 P15538 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31600356 0.83 NOTUM (0.44) NOTUMCYP11B2HTR2AHTR2CHTR2B
SCHEMBL31600663 0.79 NOTUM (0.41) NOTUMCYP11B2HTR2AHTR2CHTR2B
SCHEMBL19391610 0.76 HTR2A (0.46) NOTUMHTR2AHTR2CHTR2B
SCHEMBL3154459 0.76 CYP11B2 (0.42) NOTUMCYP11B2HTR2AHTR2CHTR2B
SCHEMBL18369759 0.74 ALDH1A1 (0.51) NOTUMCYP11B2
SCHEMBL256752 0.74 HTR2A (0.47) HTR2AHTR2CHTR2B
SCHEMBL827886 0.72 CYP11B2 (0.59) NOTUMCYP11B2CYP11B1
SCHEMBL2619231 0.70 NOTUM (1.00) NOTUM
SCHEMBL18168634 0.70 NOTUM (0.59) NOTUMCYP11B2CYP11B1
SCHEMBL13081092 0.69 HTR2A (0.46) HTR2AHTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6610692-B1 Anticoagulants MERCK & CO., INC. 2003-08-26 US disclosed
EP-1124822-A4 THROMBIN INHIBITORS MERCK & CO INC (US) 2002-04-03 EP disclosed
EP-1124822-A1 THROMBIN INHIBITORS Merck & Co., Inc. (US) 2001-08-22 EP disclosed
WO-2000026211-A1 THROMBIN INHIBITORS MERCK & CO., INC. (US) 2000-05-11 WO disclosed