SCHEMBL7215252

SCHEMBL7215252

COc1c(Cl)cc(-n2c(C)ccc2-c2ccc(S(N)(=O)=O)cc2)cc1Cl

nearest known ligand 0.53

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 17/20 0.53
PTGS1 P23219 9/20 0.53
CA12 O43570 1/20 0.46
CA1 P00915 1/20 0.46
CA2 P00918 1/20 0.46
CA9 Q16790 1/20 0.46
KDM4E B2RXH2 1/20 0.45
ALDH1A1 P00352 1/20 0.45
MAPT P10636 1/20 0.45
HPGD P15428 1/20 0.45
PTGER1 P34995 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7211995 0.89 PTGS2 (0.60) PTGS2PTGS1KDM4EALDH1A1MAPT
SCHEMBL7210291 0.87 PTGS2 (0.69) PTGS2PTGS1KDM4EALDH1A1MAPT
SCHEMBL7211987 0.85 PTGS2 (0.56) PTGS2PTGS1CA12CA1CA2
SCHEMBL7215571 0.81 PTGS2 (0.62) PTGS2PTGS1PTGER1
SCHEMBL5311980 0.80 PTGS2 (0.64) PTGS2PTGS1CA12CA1CA2
SCHEMBL5314020 0.79 CHRNA7 (0.60) PTGS2PTGS1CA12CA1CA2
SCHEMBL3026121 0.79 CHRNA7 (0.60) PTGS2PTGS1CA12CA1CA2
SCHEMBL8506105 0.79 PTGER1 (0.43) PTGS2PTGS1PTGER1
SCHEMBL7216641 0.78 PTGS2 (0.56) PTGS2PTGS1CA12CA1CA2
SCHEMBL7216779 0.77 PTGS2 (0.69) PTGS2PTGS1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1369415-A1 Substituted pyrrolyl compounds for the treatment of inflammation G.D. SEARLE & CO. (US) 2003-12-10 EP disclosed