SCHEMBL7215848

SCHEMBL7215848

CCOC(=O)c1sc2ccccc2c1N

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 7/20 0.70
MAPT P10636 7/20 0.70
ALDH1A1 P00352 6/20 0.70
KMT2A Q03164 5/20 0.70
HPGD P15428 4/20 0.70
HSD17B10 Q99714 4/20 0.70
GAA P10253 3/20 0.70
MEN1 O00255 3/20 0.70
GLA P06280 2/20 0.70
ALOX15 P16050 1/20 0.70
ATM Q13315 1/20 0.70
L3MBTL1 Q9Y468 2/20 0.63
TSHR P16473 2/20 0.63
MAPK1 P28482 1/20 0.63
LMNA P02545 3/20 0.61
IKBKB O14920 1/20 0.59
LIMK1 P53667 1/20 0.59
NOD2 Q9HC29 1/20 0.59
NPC1 O15118 2/20 0.56
RAB9A P51151 2/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31026879 1.00 KDM4E (0.70) KDM4EMAPTALDH1A1KMT2AHPGD
SCHEMBL9025206 0.84 ALDH1A1 (0.64) KDM4EMAPTALDH1A1KMT2AHPGD
SCHEMBL29513035 0.84 ALDH1A1 (0.64) KDM4EMAPTALDH1A1KMT2AHPGD
SCHEMBL9495721 0.83 LMNA (0.65) KDM4EMAPTALDH1A1KMT2AHPGD
SCHEMBL4633547 0.83 ALDH1A1 (0.63) KDM4EMAPTALDH1A1KMT2AHPGD
SCHEMBL1101766 0.83 KDM4E (1.00) KDM4EMAPTALDH1A1KMT2AHPGD
SCHEMBL30173777 0.83 KDM4E (1.00) KDM4EMAPTALDH1A1KMT2AHPGD
SCHEMBL19478160 0.81 KDM4E (0.52) KDM4EMAPTALDH1A1KMT2AHPGD
SCHEMBL9495716 0.81 ALDH1A1 (0.64) KDM4EMAPTALDH1A1KMT2AHPGD
SCHEMBL4723975 0.80 KDM4E (0.73) KDM4EMAPTALDH1A1KMT2AHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 43 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118307513-A 3-Aminobenzo [ b ] thiophene compound and preparation method and application thereof 河南工业大学 2024-07-09 CN claimed
CN-118307513-A 3-Aminobenzo [ b ] thiophene compound and preparation method and application thereof 河南工业大学 2024-07-09 CN disclosed
CN-111440216-B Synthesis method of iridium-containing complex 北京夏禾科技有限公司 2023-11-28 CN disclosed
CN-111440216-A Synthesis method of iridium-containing complex 北京夏禾科技有限公司 2020-07-24 CN disclosed
EP-2910555-B1 Organic electroluminescent materials and devices UNIVERSAL DISPLAY CORP (US) 2019-03-27 EP disclosed
EP-2910555-B1 Organic electroluminescent materials and devices UNIVERSAL DISPLAY CORP (US) 2019-03-27 EP disclosed
US-9553274-B2 Organic electroluminescent materials and devices UNIVERSAL DISPLAY CORPORATION (US) 2017-01-24 US disclosed
US-9553274-B2 Organic electroluminescent materials and devices UNIVERSAL DISPLAY CORPORATION (US) 2017-01-24 US disclosed
US-9553274-B2 Organic electroluminescent materials and devices UNIVERSAL DISPLAY CORPORATION (US) 2017-01-24 US disclosed
US-9502656-B2 Organic electroluminescent materials and devices UNIVERSAL DISPLAY CORPORATION (US) 2016-11-22 US disclosed
WO-2012131297-A1 PYRIDO [3',2' :4,5] THIENO [3, 2-D] PYRIMIDIN- 4 - YLAMINE DERIVATIVES AND THEIR THERAPEUTICAL USE BAELL JONATHAN BAYLDON (AU) 2012-10-04 WO disclosed
WO-2012131297-A1 PYRIDO [3',2' :4,5] THIENO [3, 2-D] PYRIMIDIN- 4 - YLAMINE DERIVATIVES AND THEIR THERAPEUTICAL USE BAELL JONATHAN BAYLDON (AU) 2012-10-04 WO disclosed
US-7176320-B2 Benzimidazole derivative TEIJIN LIMITED (JP) 2007-02-13 US disclosed
US-6596726-B1 Method of inhibiting epidermal growth factor by treating, with an effective inhibiting amount, a mammal, in need thereof inhibit the epidermal growth factor receptor and related receptors and, in particular, their tyrosine kinase enzyme WARNER LAMBERT COMPANY 2003-07-22 US disclosed
US-6133275-A ALPHA 1 ADRENORECEPTOR ANTAGONISTS; TREATING BENIGN PROSTATIC HYPERPLASIA AND OTHER UROLOGICAL DISEASES E.G., BLADDER OUTLET OBSTRUCTION), NEUROGENIC BLADDER AND GYNECOLOGICAL SYNDROMES, E.G., DYSMENORRHEA; UTERINE MUSCLE RELAXANTS ABBOTT LABORATORIES (US) 2000-10-17 US disclosed
EP-0808318-B1 TRICYCLIC SUBSTITUTED HEXAHYDROBENZ[E]ISOINDOLE ALPHA-1 ADRENERGIC ANTAGONISTS ABBOTT LAB (US) 2000-06-28 EP disclosed
US-5679683-A USEFUL FOR TREATING CANCER, ARTHRITIS, PSORIASIS, VASCULAR RESTENOSIS AND ANGIOGENESIS WARNER-LAMBERT COMPANY (US) 1997-10-21 US disclosed
US-5597823-A TREATING BENIGN PROSTATIC HYPERPLASIA ABBOTT LABORATORIES (US) 1997-01-28 US disclosed
EP-0741711-A1 TRICYCLIC COMPOUNDS CAPABLE OF INHIBITING TYROSINE KINASES OF THE EPIDERMAL GROWTH FACTOR RECEPTOR FAMILY WARNER-LAMBERT COMPANY (US) 1996-11-13 EP disclosed
WO-1995019970-A1 TRICYCLIC COMPOUNDS CAPABLE OF INHIBITING TYROSINE KINASES OF THE EPIDERMAL GROWTH FACTOR RECEPTOR FAMILY WARNER-LAMBERT COMPANY (US) 1995-07-27 WO disclosed