SCHEMBL7216189

SCHEMBL7216189

NS(=O)(=O)c1ccc(-n2cccc2-c2ccc(Cl)cc2)cc1

nearest known ligand 0.74

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 12/20 0.74
PTGS1 P23219 6/20 0.74
CHRNA7 P36544 2/20 0.54
CA1 P00915 6/20 0.53
CA2 P00918 6/20 0.53
CA12 O43570 4/20 0.53
CA9 Q16790 4/20 0.53
CA4 P22748 3/20 0.53
CA7 P43166 3/20 0.53
CA3 P07451 1/20 0.53
CA6 P23280 1/20 0.53
CA5A P35218 1/20 0.53
CA13 Q8N1Q1 1/20 0.53
CA14 Q9ULX7 1/20 0.53
CA5B Q9Y2D0 1/20 0.53
PDPK1 O15530 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5311727 1.00 PTGS2 (0.74) PTGS2PTGS1CHRNA7CA1CA2
SCHEMBL7212148 0.86 PTGS2 (0.76) PTGS2PTGS1CA1CA2CA12
SCHEMBL7210655 0.86 PTGS2 (0.76) PTGS2PTGS1CA1CA2CA12
SCHEMBL2463751 0.85 PTGS2 (1.00) PTGS2PTGS1CHRNA7CA1CA2
SCHEMBL7211950 0.85 PTGS2 (0.74) PTGS2PTGS1CHRNA7CA1CA2
SCHEMBL5310941 0.85 PTGS2 (0.74) PTGS2PTGS1
SCHEMBL5309601 0.85 PTGS2 (0.74) PTGS2PTGS1
SCHEMBL5308822 0.85 PTGS2 (0.74) PTGS2PTGS1CHRNA7CA1CA2
SCHEMBL5315090 0.85 PTGS2 (0.74) PTGS2PTGS1CHRNA7CA1CA2
SCHEMBL5309174 0.85 PTGS2 (1.00) PTGS2PTGS1CHRNA7CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1369415-A1 Substituted pyrrolyl compounds for the treatment of inflammation G.D. SEARLE & CO. (US) 2003-12-10 EP disclosed
EP-0946507-A1 SUBSTITUTED PYRROLYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1999-10-06 EP disclosed
WO-1998025896-A1 SUBSTITUTED PYRROLYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1998-06-18 WO disclosed