SCHEMBL7212148

SCHEMBL7212148

NS(=O)(=O)c1ccc(-n2cccc2-c2ccccc2)cc1

nearest known ligand 0.76

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 11/20 0.76
PTGS1 P23219 5/20 0.76
CA1 P00915 8/20 0.55
CA2 P00918 8/20 0.55
CA9 Q16790 8/20 0.55
CA12 O43570 5/20 0.55
PDPK1 O15530 1/20 0.48
ALDH1A1 P00352 1/20 0.48
CA5A P35218 1/20 0.48
CA5B Q9Y2D0 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7210655 0.94 PTGS2 (0.76) PTGS2PTGS1CA1CA2CA9
SCHEMBL5311727 0.86 PTGS2 (0.74) PTGS2PTGS1CA1CA2CA9
SCHEMBL5315090 0.86 PTGS2 (0.74) PTGS2PTGS1CA1CA2CA9
SCHEMBL7216189 0.86 PTGS2 (0.74) PTGS2PTGS1CA1CA2CA9
SCHEMBL7211950 0.86 PTGS2 (0.74) PTGS2PTGS1CA1CA2CA9
SCHEMBL2463751 0.86 PTGS2 (1.00) PTGS2PTGS1CA1CA2CA9
SCHEMBL5309174 0.86 PTGS2 (1.00) PTGS2PTGS1CA1CA2CA9
SCHEMBL5308822 0.86 PTGS2 (0.74) PTGS2PTGS1CA1CA2CA9
SCHEMBL7210290 0.86 PTGS2 (0.70) PTGS2PTGS1CA1CA2CA9
SCHEMBL7210285 0.86 PTGS2 (0.74) PTGS2PTGS1CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1369415-A1 Substituted pyrrolyl compounds for the treatment of inflammation G.D. SEARLE & CO. (US) 2003-12-10 EP disclosed