SCHEMBL7216664

SCHEMBL7216664

CCCOCCOc1ccc(COc2ccc3c(c2)C=C(C(=O)Nc2ccc(CN(C)C4CCOCC4)cc2)CCS3(=O)=O)cc1

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 4/20 0.47
CCR5 P51681 12/20 0.42
L3MBTL1 Q9Y468 1/20 0.36
NPC1 O15118 1/20 0.33
ALDH1A1 P00352 1/20 0.33
MAPT P10636 1/20 0.33
PKM P14618 1/20 0.33
RAB9A P51151 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
KIT P10721 1/20 0.33
FLT3 P36888 1/20 0.33
CCR7 P32248 1/20 0.33
CXCR3 P49682 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7218136 0.96 CCR2 (0.49) CCR2CCR5L3MBTL1NPC1ALDH1A1
SCHEMBL7221638 0.95 CCR2 (0.49) CCR2CCR5L3MBTL1KITFLT3
SCHEMBL7166194 0.95 CCR2 (0.49) CCR2CCR5L3MBTL1NPC1ALDH1A1
SCHEMBL3036593 0.93 CCR2 (0.56) CCR2CCR5CCR7CXCR3
SCHEMBL30227439 0.93 CCR2 (0.56) CCR2CCR5CCR7CXCR3
Hydrochloric Acid SCHEMBL7931139 0.93 CCR2 (0.55) CCR2CCR5CCR7CXCR3
SCHEMBL7222727 0.92 CCR2 (0.44) CCR2CCR5L3MBTL1SMN1; SMN2CCR7
SCHEMBL7171409 0.92 CCR2 (0.51) CCR2CCR5NPC1ALDH1A1MAPT
SCHEMBL7165818 0.91 CCR2 (0.49) CCR2CCR5L3MBTL1NPC1ALDH1A1
SCHEMBL7222634 0.91 CCR2 (0.44) CCR2CCR5L3MBTL1KITFLT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6627651-B1 Exhibiting preventive and therapeutic effects against HIV infectious diseases wherein R1 is an optionally substituted five- or six-membered ring group; X1 is a free valency or the like; W is a divalent group and inhibitors of HIV (human TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-09-30 US claimed
EP-1182195-A1 CYCLIC COMPOUNDS AND USES THEREOF Takeda Chemical Industries, Ltd. (JP) 2002-02-27 EP claimed
US-6627651-B1 Exhibiting preventive and therapeutic effects against HIV infectious diseases wherein R1 is an optionally substituted five- or six-membered ring group; X1 is a free valency or the like; W is a divalent group and inhibitors of HIV (human TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-09-30 US disclosed
EP-1182195-A1 CYCLIC COMPOUNDS AND USES THEREOF Takeda Chemical Industries, Ltd. (JP) 2002-02-27 EP disclosed