SCHEMBL7166194

SCHEMBL7166194

CCCOCc1ccc(COc2ccc3c(c2)C=C(C(=O)Nc2ccc(CN(C)C4CCOCC4)cc2)CCS3(=O)=O)cc1

nearest known ligand 0.49

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 6/20 0.49
CCR5 P51681 11/20 0.43
L3MBTL1 Q9Y468 1/20 0.34
CXCR3 P49682 3/20 0.34
CCR7 P32248 2/20 0.34
CXCR5 P32302 1/20 0.33
NPC1 O15118 1/20 0.33
ALDH1A1 P00352 1/20 0.33
MAPT P10636 1/20 0.33
PKM P14618 1/20 0.33
RAB9A P51151 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7216664 0.95 CCR2 (0.47) CCR2CCR5L3MBTL1CXCR3CCR7
SCHEMBL7218136 0.95 CCR2 (0.49) CCR2CCR5L3MBTL1CXCR3CCR7
SCHEMBL7171409 0.92 CCR2 (0.51) CCR2CCR5CXCR3CCR7CXCR5
SCHEMBL7222495 0.92 CCR2 (0.46) CCR2CCR5L3MBTL1CXCR3CCR7
SCHEMBL7221638 0.92 CCR2 (0.49) CCR2CCR5L3MBTL1CXCR3CCR7
SCHEMBL7167251 0.91 CCR2 (0.47) CCR2CCR5L3MBTL1CXCR3CXCR5
SCHEMBL7215854 0.91 CCR2 (0.51) CCR2CCR5CXCR3CCR7NPC1
SCHEMBL7165818 0.90 CCR2 (0.49) CCR2CCR5L3MBTL1CXCR3CCR7
SCHEMBL7222727 0.90 CCR2 (0.44) CCR2CCR5L3MBTL1CXCR3CCR7
SCHEMBL7216597 0.90 CCR2 (0.48) CCR2CCR5L3MBTL1CXCR3CCR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6627651-B1 Exhibiting preventive and therapeutic effects against HIV infectious diseases wherein R1 is an optionally substituted five- or six-membered ring group; X1 is a free valency or the like; W is a divalent group and inhibitors of HIV (human TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-09-30 US disclosed
US-20030078189-A1 Medicinal compositions for oral use TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2003-04-24 US disclosed
EP-1236476-A1 MEDICINAL COMPOSITIONS FOR ORAL USE Takeda Chemical Industries, Ltd. (JP) 2002-09-04 EP disclosed
EP-1182195-A1 CYCLIC COMPOUNDS AND USES THEREOF Takeda Chemical Industries, Ltd. (JP) 2002-02-27 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030078189-A1 Medicinal compositions for oral use CCR5, CXCR3, CCL5 CCR2 23/4885CCR5 1/4885L3MBTL1 3426/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.