SCHEMBL7216679

SCHEMBL7216679

CCCN(CCC)C(=O)Cn1c(=O)[nH]c2cnc(-c3ccc(Cl)cc3)nc21

nearest known ligand 0.52

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 1/20 0.51
USP1 O94782 7/20 0.44
TSPO P30536 3/20 0.42
GMNN O75496 1/20 0.41
LMNA P02545 1/20 0.41
POLB P06746 1/20 0.41
CYP3A4 P08684 1/20 0.41
BLM P54132 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7215568 0.90 ADORA3 (0.55) ADORA3USP1TSPO
SCHEMBL2210780 0.72 ADORA3 (0.62) ADORA3USP1
SCHEMBL7210740 0.71 TSPO (0.62) TSPO
SCHEMBL7210956 0.70 ADORA3 (0.65) ADORA3USP1CYP3A4
SCHEMBL7215331 0.70 ADORA3 (0.68) ADORA3USP1
SCHEMBL7210455 0.69 TSPO (0.77) USP1TSPO
SCHEMBL9692288 0.68
SCHEMBL4147487 0.68 ADORA3 (0.56) ADORA3USP1
SCHEMBL7210798 0.68 TSPO (0.88) USP1TSPO
SCHEMBL10387488 0.68 GMNN (0.44) TSPOGMNNLMNAPOLBCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1036794-B1 2-ARYL-8-OXODIHYDROPURINE DERIVATIVES, PROCESS FOR PRODUCING THE SAME, MEDICINAL COMPOSITIONS CONTAINING THE SAME, AND INTERMEDIATES THEREOF DAINIPPON PHARMACEUTICAL CO (JP) 2003-08-27 EP disclosed
US-6372740-B1 NERVOUS SYSTEM DISORDERS, ANTIEPILEPTIC AGENTS AND ANTIDEPRESSANTS DAINIPPON PHARMACEUTICAL CO., LTD. (JP) 2002-04-16 US disclosed
EP-1036794-A1 2-ARYL-8-OXODIHYDROPURINE DERIVATIVES, PROCESS FOR PRODUCING THE SAME, MEDICINAL COMPOSITIONS CONTAINING THE SAME, AND INTERMEDIATES THEREOF Dainippon Pharmaceutical Co., Ltd. (JP) 2000-09-20 EP disclosed