SCHEMBL7217322

SCHEMBL7217322

CCn1c(=O)[nH]c2nc[nH]c2c1=O.[KH]

nearest known ligand 0.97

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 11/20 0.97
PDE4A P27815 9/20 0.97
PDE4B Q07343 9/20 0.97
PDE4C Q08493 9/20 0.97
PDE4D Q08499 9/20 0.97
ADORA2B P29275 14/20 0.75
ADORA3 P0DMS8 8/20 0.75
HPGD P15428 1/20 0.47
ADORA1 P30542 1/20 0.47
BLM P54132 1/20 0.47
PDE3A Q14432 1/20 0.47
HSD17B10 Q99714 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL380135 0.98 ADORA2A (1.00) ADORA2APDE4APDE4BPDE4CPDE4D
SCHEMBL27396492 0.98 ADORA2A (1.00) ADORA2APDE4APDE4BPDE4CPDE4D
SCHEMBL4423680 0.86 ADORA2B (1.00) ADORA2APDE4APDE4BPDE4CPDE4D
SCHEMBL6233166 0.83 ADORA2B (1.00) ADORA2APDE4APDE4BPDE4CPDE4D
SCHEMBL27395394 0.83 ADORA2B (1.00) ADORA2APDE4APDE4BPDE4CPDE4D
SCHEMBL5515444 0.82 ADORA2A (0.71) ADORA2APDE4APDE4BPDE4CPDE4D
SCHEMBL27586849 0.82 ADORA2A (0.71) ADORA2APDE4APDE4BPDE4CPDE4D
SCHEMBL7455767 0.82 ADORA2A (0.71) ADORA2APDE4APDE4BPDE4CPDE4D
SCHEMBL1892011 0.82 ADORA2B (0.92) ADORA2APDE4APDE4BPDE4CPDE4D
SCHEMBL60158 0.81 ADORA2A (0.70) ADORA2APDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6566384-B1 For therapy of cancer, inflammation and inflammatory diseases, tissue degeneration, periodontal disease, ophthalmological disease, dermatological disorders, fever, cardiovascular effects, haemorrhage, coagulation and acute phase response DARWIN DISCOVERY LTD. (GB) 2003-05-20 US disclosed