SCHEMBL7220061

SCHEMBL7220061

O=C(O)C=CC(=O)Nc1cc2c(Nc3ccc(F)c(Cl)c3)ncnc2cn1

nearest known ligand 0.79

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
EGFR P00533 19/20 0.79
ERBB2 P04626 16/20 0.79
ERBB4 Q15303 12/20 0.74
JAK3 P52333 3/20 0.70
MEN1 O00255 1/20 0.68
KMT2A Q03164 1/20 0.68
GRM1 Q13255 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4184896 0.89 EGFR (0.78) EGFRERBB2ERBB4JAK3MEN1
SCHEMBL2993868 0.88 EGFR (1.00) EGFRERBB2ERBB4JAK3MEN1
SCHEMBL7219678 0.87 EGFR (0.64) EGFRERBB2ERBB4JAK3
SCHEMBL7216169 0.86 EGFR (0.63) EGFRERBB2ERBB4JAK3
SCHEMBL4187462 0.84 EGFR (0.75) EGFRERBB2ERBB4JAK3MEN1
SCHEMBL238877 0.81 EGFR (1.00) EGFRERBB2ERBB4JAK3MEN1
SCHEMBL29409571 0.81 EGFR (1.00) EGFRERBB2ERBB4JAK3MEN1
SCHEMBL7242341 0.81 EGFR (0.53) EGFRERBB2ERBB4JAK3MEN1
SCHEMBL4350856 0.80 EGFR (0.75) EGFRERBB2ERBB4JAK3MEN1
SCHEMBL7238659 0.80 EGFR (0.76) EGFRERBB2ERBB4JAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6602863-B1 Irreversible inhibitors of tyrosine kinases WARNER-LAMBERT COMPANY 2003-08-05 US claimed
US-6602863-B1 Irreversible inhibitors of tyrosine kinases WARNER-LAMBERT COMPANY 2003-08-05 US disclosed