SCHEMBL7221507

SCHEMBL7221507

Cc1ccc(-c2ccc3cc(C(=O)Nc4ccc(CN(C)C5CCOCC5)cc4)n(C)c3c2)cc1

nearest known ligand 0.59

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 6/20 0.59
THRB P10828 1/20 0.46
CCR5 P51681 6/20 0.45
HDAC1 Q13547 1/20 0.44
MCHR1 Q99705 1/20 0.42
CCR7 P32248 2/20 0.41
CXCR3 P49682 2/20 0.41
MAPT P10636 3/20 0.40
LMNA P02545 1/20 0.40
PTGDR2 Q9Y5Y4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13148497 0.86 CCR5 (0.50) CCR2THRBCCR5HDAC1MCHR1
SCHEMBL7216354 0.82 CCR2 (0.61) CCR2CCR5HDAC1MCHR1CCR7
SCHEMBL7218106 0.81 CCR2 (0.61) CCR2CCR5HDAC1MCHR1CCR7
SCHEMBL5204989 0.78 CCR2 (0.59) CCR2CCR5HDAC1MCHR1CCR7
SCHEMBL5209524 0.76 CCR2 (0.73) CCR2CCR5CCR7CXCR3
SCHEMBL5209267 0.76 CCR2 (0.55) CCR2CCR5HDAC1MCHR1
SCHEMBL5205096 0.75 CCR2 (0.72) CCR2CCR5
SCHEMBL5203761 0.75 CCR2 (0.72) CCR2CCR5HDAC1CCR7CXCR3
SCHEMBL3026537 0.75 CCR2 (0.77) CCR2CCR5
SCHEMBL5204966 0.75 CCR2 (1.00) CCR2CCR5CCR7CXCR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6627651-B1 Exhibiting preventive and therapeutic effects against HIV infectious diseases wherein R1 is an optionally substituted five- or six-membered ring group; X1 is a free valency or the like; W is a divalent group and inhibitors of HIV (human TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-09-30 US disclosed
EP-1182195-A1 CYCLIC COMPOUNDS AND USES THEREOF Takeda Chemical Industries, Ltd. (JP) 2002-02-27 EP disclosed