SCHEMBL7223087

SCHEMBL7223087

C=C[C@@H](c1cccc(F)c1)C(C(=O)O)C(=O)O

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 1/20 0.45
HDAC7 Q8WUI4 1/20 0.45
HDAC5 Q9UQL6 1/20 0.45
CES2 O00748 2/20 0.44
CES1 P23141 2/20 0.44
CNR2 P34972 1/20 0.41
EPHX1 P07099 1/20 0.39
IDO1 P14902 1/20 0.38
TDO2 P48775 1/20 0.38
MTOR P42345 1/20 0.38
KDM4E B2RXH2 1/20 0.38
SLC1A1 P43005 1/20 0.37
LMNA P02545 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7223081 1.00 HDAC4 (0.45) HDAC4HDAC7HDAC5CES2CES1
SCHEMBL7218494 0.82 HDAC4 (0.44) HDAC4HDAC7HDAC5CES2CES1
SCHEMBL7218493 0.82 HDAC4 (0.44) HDAC4HDAC7HDAC5CES2CES1
SCHEMBL5836538 0.81 LMNA (0.51) HDAC4HDAC7HDAC5CES2CES1
SCHEMBL27843791 0.74 HDAC4 (0.51) HDAC4HDAC7HDAC5CES2CES1
SCHEMBL3711116 0.73 SRC (0.58) HDAC4HDAC7HDAC5CES2CES1
SCHEMBL7216851 0.73 HDAC4 (0.44) HDAC4HDAC7HDAC5CES2CES1
SCHEMBL4022595 0.73 CYP2C19 (0.68) HDAC4HDAC7HDAC5CES2CES1
SCHEMBL287924 0.72 CES2 (0.66) HDAC4HDAC7HDAC5CES2CES1
SCHEMBL4390797 0.72 HDAC4 (0.53) HDAC4HDAC7HDAC5CES2CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6593346-B2 Substituted 3-(piperidin-1-ylmethyl)cyclopentylamines, useful as modulators of the chemokine receptors CCR-5 and/or CC R-3. MERCK & CO. INC. 2003-07-15 US disclosed
US-6358979-B1 FOR THERAPY AND PROPHYLAXIS OF ASTHMA, ALLERGIC RHINITIS, DERMATITIS, CONJUNCTIVITIS, ATHEROSCLEROSIS OR RHEUMATOID ARTHRITIS, INFECTION BY HIV, TREATING INFECTION BY HIV, DELAYING OF THE ONSET OF AIDS MERCK & CO., INC. 2002-03-19 US disclosed