SCHEMBL7223276

SCHEMBL7223276

CCOc1cc2c(cc1OCC)CC(C(=O)OCc1ccccc1)NC2

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.45
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
KDM4E B2RXH2 2/20 0.42
HSD17B10 Q99714 2/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
MAPK1 P28482 1/20 0.42
CYP2C19 P33261 1/20 0.42
ACE P12821 1/20 0.41
GAA P10253 1/20 0.41
MAPK10 P53779 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
LMNA P02545 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.40
HDAC8 Q9BY41 2/20 0.40
BACE1 P56817 1/20 0.40
MRGPRX4 Q96LA9 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7223266 1.00 TSHR (0.45) TSHRMEN1KMT2AKDM4EHSD17B10
SCHEMBL7225047 0.88 ACE (0.47) TSHRMEN1KMT2AACESMN1; SMN2
SCHEMBL7225043 0.88 ACE (0.47) TSHRMEN1KMT2AACESMN1; SMN2
SCHEMBL8235210 0.81 KMT2A (0.53) TSHRMEN1KMT2AMAPK1L3MBTL1
SCHEMBL7677497 0.81 KMT2A (0.53) TSHRMEN1KMT2AMAPK1L3MBTL1
SCHEMBL27627519 0.81 KMT2A (0.53) TSHRMEN1KMT2AMAPK1L3MBTL1
SCHEMBL243337 0.81 AGTR2 (0.50) SMN1; SMN2HDAC8
Hydrochloric Acid SCHEMBL10755389 0.80 MEN1 (0.55) TSHRMEN1KMT2AKDM4EHSD17B10
SCHEMBL7221112 0.80 ACHE (0.42) TSHRMEN1KMT2AKDM4EHSD17B10
SCHEMBL7221115 0.80 ACHE (0.42) TSHRMEN1KMT2AKDM4EHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003101967-A1 PREPARATION OF CHIRAL 1,2,3,4-TETRAHYDRO-6,7-DIALKOXY-3-ISOQUINOLINECARBOXYLIC ACID AND DERIVATIVES BY REACTING LEVODOPA WITH FORMALDEHYDE OR FORMALDEHYDE PRECURSORS APTEX PHARMACHEM INC. (CA) 2003-12-11 WO claimed
US-6642384-B1 Forming intermediate to moexipril; cyclizing levodopa with formaldehyde; protecting amine, alkylating phenols, esterifying carboxylic acid and optionally deprotecting BRANTFORD CHEMICALS INC. (CA) 2003-11-04 US claimed