SCHEMBL7224299

SCHEMBL7224299

Cc1ccc(-c2ccc(C(=O)N[C@@H]3C[C@H]4CC[C@@H]3N4)s2)s1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.45
RAB9A P51151 2/20 0.45
CHRNA7 P36544 10/20 0.39
HTR3E A5X5Y0 5/20 0.39
HTR3B O95264 5/20 0.39
HTR3A P46098 5/20 0.39
HTR3D Q70Z44 5/20 0.39
HTR3C Q8WXA8 5/20 0.39
TAS1R3 Q7RTX0 1/20 0.39
TAS1R1 Q7RTX1 1/20 0.39
F10 P00742 1/20 0.39
ESR1 P03372 1/20 0.37
ESRRG P62508 1/20 0.37
ESR2 Q92731 1/20 0.37
PTPN1 P18031 1/20 0.37
PTPN11 Q06124 1/20 0.37
KDM4E B2RXH2 1/20 0.37
TP53 P04637 1/20 0.37
MAPT P10636 1/20 0.37
HPGD P15428 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7223510 0.93 NPC1 (0.52) NPC1RAB9ACHRNA7TAS1R3TAS1R1
Hydrochloric Acid SCHEMBL7231904 0.91 NPC1 (0.51) NPC1RAB9ACHRNA7TAS1R3TAS1R1
SCHEMBL7232814 0.88 CHRNA7 (0.37) NPC1RAB9ACHRNA7HTR3EHTR3B
SCHEMBL7230458 0.87 NPC1 (0.38) NPC1RAB9ACHRNA7HTR3EHTR3B
SCHEMBL7224991 0.86 ESRRG (0.46) NPC1RAB9ACHRNA7HTR3EHTR3B
SCHEMBL7224322 0.86 CHRNA7 (0.40) RAB9ACHRNA7HTR3EHTR3BHTR3A
SCHEMBL7226078 0.85 NPC1 (0.38) NPC1RAB9ACHRNA7HTR3EHTR3B
SCHEMBL7231162 0.85 NPC1 (0.43) NPC1RAB9ATAS1R3TAS1R1F10
SCHEMBL7225345 0.85 CHRNA7 (0.41) CHRNA7HTR3EHTR3BHTR3AHTR3D
SCHEMBL7232316 0.85 NPC1 (0.43) NPC1RAB9ATAS1R3TAS1R1F10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US claimed
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US disclosed