SCHEMBL7230458

SCHEMBL7230458

Cc1cnc(-c2ccc(C(=O)N[C@@H]3C[C@H]4CC[C@@H]3N4)s2)s1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.38
RAB9A P51151 3/20 0.38
KDM4E B2RXH2 1/20 0.38
TP53 P04637 1/20 0.38
MAPT P10636 1/20 0.38
HPGD P15428 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
HSD17B10 Q99714 1/20 0.38
CHRNA7 P36544 8/20 0.37
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
HTR3E A5X5Y0 5/20 0.35
HTR3B O95264 5/20 0.35
HTR3A P46098 5/20 0.35
HTR3D Q70Z44 5/20 0.35
HTR3C Q8WXA8 5/20 0.35
AKT1 P31749 2/20 0.35
MAPK13 O15264 1/20 0.34
MAPK12 P53778 1/20 0.34
MAPK11 Q15759 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7223422 0.88 HPGD (0.38) NPC1RAB9AKDM4ETP53MAPT
SCHEMBL7224906 0.87 CHRNA7 (0.38) NPC1RAB9AKDM4ETP53MAPT
SCHEMBL7224299 0.87 NPC1 (0.45) NPC1RAB9AKDM4ETP53MAPT
SCHEMBL7232814 0.84 CHRNA7 (0.37) NPC1RAB9ACHRNA7HTR3EHTR3B
SCHEMBL7226078 0.84 NPC1 (0.38) NPC1RAB9AKDM4ETP53MAPT
SCHEMBL7223147 0.83 HDAC1 (0.41) NPC1RAB9AKDM4ETP53MAPT
SCHEMBL7227405 0.83 MAPK13 (0.50) KDM4ECHRNA7HTR3EHTR3BHTR3A
SCHEMBL7230264 0.83 CHRNA7 (0.40) NPC1RAB9AKDM4ETP53MAPT
SCHEMBL7230597 0.82 NPC1 (0.39) NPC1RAB9AKDM4ETP53MAPT
SCHEMBL7223510 0.82 NPC1 (0.52) NPC1RAB9ACHRNA7MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US claimed
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US disclosed