SCHEMBL7224305

SCHEMBL7224305

Cc1ccc(-c2cnc(C(=O)N[C@@H]3C[C@H]4CC[C@@H]3N4)o2)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 4/20 0.46
HDAC6 Q9UBN7 4/20 0.46
CA12 O43570 2/20 0.45
CA1 P00915 2/20 0.45
CA2 P00918 2/20 0.45
CA4 P22748 2/20 0.45
SLC6A2 P23975 1/20 0.42
SLC6A4 P31645 1/20 0.42
SLC6A3 Q01959 1/20 0.42
NPC1 O15118 3/20 0.37
RAB9A P51151 3/20 0.37
KMT2A Q03164 3/20 0.36
MEN1 O00255 1/20 0.36
S1PR1 P21453 1/20 0.36
CNR1 P21554 1/20 0.36
TUBB4A P04350 1/20 0.36
TUBB P07437 1/20 0.36
TUBA3C P0DPH7 1/20 0.36
TUBA1B P68363 1/20 0.36
TUBA4A P68366 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7226687 0.90 TUBB4A (0.46) HDAC1HDAC6CA12CA1CA2
SCHEMBL7231845 0.90 CA12 (0.44) HDAC1HDAC6CA12CA1CA2
SCHEMBL7222561 0.89 CA12 (0.48) HDAC1HDAC6CA12CA1CA2
SCHEMBL7231985 0.89 HDAC1 (0.46) HDAC1HDAC6CA12CA1CA2
SCHEMBL7226619 0.89 HDAC1 (0.46) HDAC1HDAC6CA12CA1CA2
SCHEMBL7234526 0.89 HDAC1 (0.47) HDAC1HDAC6CA12CA1CA2
SCHEMBL7073214 0.89 TUBB4A (0.47) HDAC1HDAC6CA12CA1CA2
SCHEMBL7232218 0.89 HDAC6 (0.48) HDAC1HDAC6CA12CA1CA2
SCHEMBL7234556 0.88 CA12 (0.44) HDAC1HDAC6CA12CA1CA2
Hydrochloric Acid SCHEMBL7072564 0.88 TUBB4A (0.46) HDAC1HDAC6CA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US claimed
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US disclosed