SCHEMBL7224563

SCHEMBL7224563

CC(=O)c1ccc(-c2ccc(C(=O)N[C@@H]3C[C@H]4CC[C@@H]3N4)s2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 2/20 0.49
PTPN11 Q06124 2/20 0.49
CHRNA7 P36544 5/20 0.45
HTR3E A5X5Y0 4/20 0.45
HTR3B O95264 4/20 0.45
HTR3A P46098 4/20 0.45
HTR3D Q70Z44 4/20 0.45
HTR3C Q8WXA8 4/20 0.45
HDAC6 Q9UBN7 1/20 0.44
ESR1 P03372 1/20 0.44
ESRRG P62508 1/20 0.44
ESR2 Q92731 1/20 0.44
MAPK11 Q15759 10/20 0.40
MAPK14 Q16539 10/20 0.40
MAPK13 O15264 1/20 0.39
MAPK12 P53778 1/20 0.39
KDM4E B2RXH2 1/20 0.38
NPC1 O15118 1/20 0.38
ALDH1A1 P00352 1/20 0.38
HPGD P15428 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7232261 0.90 CHRNA7 (0.47) PTPN1PTPN11CHRNA7HTR3EHTR3B
SCHEMBL7223923 0.89 PTPN11 (0.49) PTPN1PTPN11CHRNA7HTR3EHTR3B
SCHEMBL7224991 0.89 ESRRG (0.46) PTPN1PTPN11CHRNA7HTR3EHTR3B
SCHEMBL7230658 0.87 CHRNA7 (0.46) PTPN1PTPN11CHRNA7HTR3EHTR3B
SCHEMBL7231972 0.87 ESRRG (0.46) PTPN1PTPN11CHRNA7HTR3EHTR3B
SCHEMBL375517 0.86 CHRNA7 (0.57) PTPN1PTPN11CHRNA7HTR3EHTR3B
SCHEMBL7223338 0.86 CHRNA7 (0.57) PTPN1PTPN11CHRNA7HTR3EHTR3B
SCHEMBL7224860 0.86 KDM4E (0.55) PTPN1PTPN11CHRNA7HTR3EHTR3B
SCHEMBL7232519 0.85 MAPK11 (0.48) PTPN1PTPN11CHRNA7HTR3EHTR3B
SCHEMBL7224193 0.84 HDAC3 (0.53) PTPN1PTPN11CHRNA7HTR3EHTR3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US claimed
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US disclosed