SCHEMBL7224860

SCHEMBL7224860

COc1ccc(-c2ccc(C(=O)N[C@@H]3C[C@H]4CC[C@@H]3N4)s2)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.55
SMN1; SMN2 Q16637 2/20 0.55
NPC1 O15118 1/20 0.55
ALDH1A1 P00352 1/20 0.55
GLA P06280 1/20 0.55
GAA P10253 1/20 0.55
MAPT P10636 1/20 0.55
HPGD P15428 1/20 0.55
LMNA P02545 1/20 0.53
MAPK11 Q15759 1/20 0.48
MAPK14 Q16539 1/20 0.48
ESR1 P03372 1/20 0.43
ESRRG P62508 1/20 0.43
ESR2 Q92731 1/20 0.43
PTPN1 P18031 1/20 0.43
PTPN11 Q06124 1/20 0.43
CHRNA7 P36544 6/20 0.42
HTR3E A5X5Y0 4/20 0.42
HTR3B O95264 4/20 0.42
HTR3A P46098 4/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7232229 0.90 HDAC6 (0.50) KDM4ESMN1; SMN2NPC1ALDH1A1GLA
SCHEMBL7224991 0.88 ESRRG (0.46) KDM4ENPC1ALDH1A1HPGDMAPK11
SCHEMBL7224563 0.86 PTPN1 (0.49) KDM4ENPC1ALDH1A1HPGDMAPK11
SCHEMBL7224866 0.86 CTSC (0.40) KDM4ESMN1; SMN2NPC1ALDH1A1GLA
SCHEMBL7225220 0.86 CHRNA7 (0.39) KDM4ESMN1; SMN2NPC1ALDH1A1GLA
SCHEMBL7231972 0.86 ESRRG (0.46) MAPK11MAPK14ESR1ESRRGESR2
SCHEMBL375517 0.85 CHRNA7 (0.57) KDM4ESMN1; SMN2NPC1ALDH1A1MAPT
SCHEMBL7223338 0.85 CHRNA7 (0.57) KDM4ESMN1; SMN2NPC1ALDH1A1MAPT
SCHEMBL7225149 0.85 HTR4 (0.37) KDM4ESMN1; SMN2NPC1ALDH1A1GLA
SCHEMBL7225345 0.85 CHRNA7 (0.41) CHRNA7HTR3EHTR3BHTR3AHTR3D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US claimed
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US disclosed