SCHEMBL7225955

SCHEMBL7225955

O=C(N[C@@H]1C[C@H]2CC[C@@H]1N2)c1ccc(-c2ccccc2-c2ccco2)o1

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.40
RAB9A P51151 4/20 0.40
ALDH1A1 P00352 2/20 0.40
KDM4E B2RXH2 1/20 0.39
NPSR1 Q6W5P4 2/20 0.37
LMNA P02545 1/20 0.37
GAA P10253 1/20 0.37
HTT P42858 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
TSHR P16473 1/20 0.36
HTR3E A5X5Y0 1/20 0.35
HTR3B O95264 1/20 0.35
HTR3A P46098 1/20 0.35
HTR3D Q70Z44 1/20 0.35
HTR3C Q8WXA8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7224316 0.88 NPC1 (0.42) NPC1RAB9AALDH1A1KDM4ENPSR1
SCHEMBL7226523 0.86 SMN1; SMN2 (0.42) NPC1RAB9AALDH1A1KDM4ENPSR1
SCHEMBL7234830 0.86 RAB9A (0.42) NPC1RAB9ANPSR1LMNAGAA
SCHEMBL7223990 0.86 RAB9A (0.42) NPC1RAB9AALDH1A1KDM4ENPSR1
SCHEMBL7223992 0.86 RAB9A (0.42) NPC1RAB9AALDH1A1KDM4ENPSR1
SCHEMBL7234111 0.85 NPC1 (0.37) NPC1RAB9AALDH1A1KDM4ENPSR1
SCHEMBL7072612 0.85 RAB9A (0.49) NPC1RAB9AALDH1A1KDM4ENPSR1
SCHEMBL7225840 0.85 RAB9A (0.41) NPC1RAB9AALDH1A1KDM4ENPSR1
SCHEMBL7231145 0.85 SLC9A1 (0.44) NPC1RAB9ANPSR1LMNAGAA
SCHEMBL7226764 0.85 RAB9A (0.53) NPC1RAB9AALDH1A1KDM4ENPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US claimed
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US disclosed