SCHEMBL7225979

SCHEMBL7225979

O=C(N[C@@H]1C[C@H]2CC[C@@H]1N2)c1ccc(-c2ccc(NC(=O)C(F)(F)F)cc2)s1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 5/20 0.41
HTR3E A5X5Y0 4/20 0.41
HTR3B O95264 4/20 0.41
HTR3A P46098 4/20 0.41
HTR3D Q70Z44 4/20 0.41
HTR3C Q8WXA8 4/20 0.41
ESRRG P62508 7/20 0.41
PTPN11 Q06124 3/20 0.41
PTPN2 P17706 1/20 0.41
ESR1 P03372 2/20 0.40
PTPN1 P18031 2/20 0.40
ESR2 Q92731 1/20 0.40
KDM4E B2RXH2 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
MEN1 O00255 1/20 0.39
MAPT P10636 1/20 0.39
KMT2A Q03164 1/20 0.39
LMNA P02545 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7224673 0.92 CHRNA7 (0.44) CHRNA7HTR3EHTR3BHTR3AHTR3D
SCHEMBL7226094 0.87 CHRNA7 (0.42) CHRNA7HTR3EHTR3BHTR3AHTR3D
SCHEMBL7230658 0.87 CHRNA7 (0.46) CHRNA7HTR3EHTR3BHTR3AHTR3D
SCHEMBL7224429 0.86 MAPK11 (0.48) CHRNA7HTR3EHTR3BHTR3AHTR3D
SCHEMBL7224594 0.85 CHRNA7 (0.40) CHRNA7HTR3EHTR3BHTR3AHTR3D
SCHEMBL7232742 0.85 F10 (0.32) CHRNA7SMN1; SMN2NPC1RAB9AMEN1
SCHEMBL7222908 0.84 EPHX2 (0.34) KDM4ESMN1; SMN2MAPT
SCHEMBL7223409 0.84 PTPN11 (0.44) PTPN11PTPN1NPC1RAB9AMEN1
SCHEMBL7223114 0.83 CHRNA7 (0.40) CHRNA7HTR3EHTR3BHTR3AHTR3D
SCHEMBL6488520 0.82 CHRNA7 (0.44) CHRNA7HTR3EHTR3BHTR3AHTR3D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US claimed
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US disclosed