SCHEMBL7223409

SCHEMBL7223409

O=C(N[C@@H]1C[C@H]2CC[C@@H]1N2)c1cnc(-c2ccc(NC(=O)C(F)(F)F)cc2)s1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN11 Q06124 1/20 0.44
PTPN1 P18031 1/20 0.41
SLC6A3 Q01959 1/20 0.38
KCNH2 Q12809 1/20 0.38
TAAR1 Q96RJ0 1/20 0.38
USP30 Q70CQ3 1/20 0.38
HDAC1 Q13547 4/20 0.37
HDAC6 Q9UBN7 4/20 0.37
TP53 P04637 2/20 0.37
ULK1 O75385 1/20 0.36
PPARA Q07869 1/20 0.35
HDAC3 O15379 3/20 0.35
HDAC4 P56524 3/20 0.35
HDAC7 Q8WUI4 3/20 0.35
HDAC2 Q92769 3/20 0.35
HDAC10 Q969S8 3/20 0.35
HDAC11 Q96DB2 3/20 0.35
HDAC8 Q9BY41 3/20 0.35
HDAC9 Q9UKV0 3/20 0.35
HDAC5 Q9UQL6 3/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7230386 0.90 USP30 (0.38) PTPN11PTPN1SLC6A3KCNH2TAAR1
SCHEMBL7232579 0.88 PTPN11 (0.43) PTPN11PTPN1SLC6A3KCNH2TAAR1
SCHEMBL7232029 0.86 HDAC1 (0.49) PTPN11PTPN1USP30HDAC1HDAC6
SCHEMBL7226045 0.85 USP30 (0.43) PTPN11PTPN1SLC6A3KCNH2TAAR1
SCHEMBL7226143 0.85 PTPN11 (0.49) PTPN11PTPN1SLC6A3USP30HDAC1
SCHEMBL7224996 0.84 USP30 (0.42) PTPN11PTPN1SLC6A3KCNH2TAAR1
SCHEMBL7225979 0.84 CHRNA7 (0.41) PTPN11PTPN1KCNH2MEN1NPC1
SCHEMBL7223360 0.84 MAPK11 (0.39) USP30HDAC1HDAC6ULK1HDAC3
SCHEMBL7223371 0.83 USP30 (0.42) PTPN11PTPN1SLC6A3KCNH2TAAR1
SCHEMBL7234180 0.83 USP30 (0.42) PTPN11PTPN1SLC6A3KCNH2TAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US claimed
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US disclosed