SCHEMBL7227808

SCHEMBL7227808

CCCCS(=O)(=O)NC(Cc1ccc(OCC2CN(c3ccc(C#N)cc3)C(=O)O2)cc1)C(=O)OC

nearest known ligand 0.49

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 13/20 0.49
ITGB3 P05106 5/20 0.45
ITGA2B P08514 5/20 0.45
ITGAV P06756 1/20 0.45
CHRM2 P08172 1/20 0.45
SLC6A4 P31645 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7235026 0.91 GRM2 (0.55) GRM2ITGB3ITGA2BITGAVCHRM2
SCHEMBL7236076 0.89 ITGB3 (0.50) GRM2ITGB3ITGA2BITGAVCHRM2
SCHEMBL7236747 0.87 GRM2 (0.49) GRM2ITGB3ITGA2BITGAVCHRM2
SCHEMBL7228244 0.85 GRM2 (0.50) GRM2
SCHEMBL7241085 0.84 ITGB3 (0.48) GRM2ITGB3ITGA2BITGAVCHRM2
SCHEMBL7234939 0.84 ITGB3 (0.46) GRM2ITGB3ITGA2BITGAVCHRM2
SCHEMBL7392208 0.83 ITGB3 (0.44) GRM2ITGB3ITGA2BITGAVCHRM2
SCHEMBL3267022 0.83 ITGB3 (0.57) GRM2ITGB3ITGA2BITGAVCHRM2
SCHEMBL7235820 0.81 ITGB3 (0.44) GRM2ITGB3ITGA2BITGAVCHRM2
SCHEMBL7229264 0.81 GRM2 (0.47) GRM2ITGB3ITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6602876-B1 Adhesion receptor antagonists MERCK PATENT GMBH (DE) 2003-08-05 US disclosed
US-6204280-B1 OXAZOLIDINONE DERIVATIVE, ANTICOAGULANT MERCK PATENT GESELLSCHAFT MIT BERSCHRANKTER HAFTUNG (DE) 2001-03-20 US disclosed
EP-0710657-B1 Antagonists of adhesion receptors MERCK PATENT GMBH (DE) 1998-08-26 EP disclosed
EP-0710657-A1 Antagonists of adhesion receptors MERCK PATENT GmbH (DE) 1996-05-08 EP disclosed