SCHEMBL722817

SCHEMBL722817

O=C(N1CCc2cc3ccc(Cl)nc3cc2CC1)C(F)(F)F

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 7/20 0.51
ESR2 Q92731 7/20 0.51
SMN1; SMN2 Q16637 1/20 0.41
ABHD6 Q9BV23 2/20 0.38
CYP11B2 P19099 1/20 0.37
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
HDAC6 Q9UBN7 1/20 0.34
HPGD P15428 2/20 0.34
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA7 P43166 1/20 0.34
CA9 Q16790 1/20 0.34
DRD2 P14416 1/20 0.34
MAPT P10636 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL722449 0.82 ESR1 (0.48) ESR1ESR2SMN1; SMN2CYP11B2HPGD
Trifluoroacetic Acid SCHEMBL719783 0.76 KDM1A (0.39) DRD2
SCHEMBL719748 0.76 ESR1 (0.52) ESR1ESR2ABHD6CYP11B2HDAC6
SCHEMBL719099 0.75 DRD2 (0.44) MEN1KMT2ADRD2
SCHEMBL2585109 0.75 ESR1 (0.62) ESR1ESR2ABHD6HDAC6
SCHEMBL373697 0.73 ESR2 (0.83) ESR1ESR2ABHD6HDAC6CA1
SCHEMBL3715395 0.71 ESR1 (0.48) ESR1ESR2ABHD6CYP11B2HDAC6
SCHEMBL719752 0.71 ESR1 (0.48) ESR1ESR2SMN1; SMN2KMT2ADRD2
SCHEMBL719456 0.70 ESR1 (0.56) ESR1ESR2ABHD6CYP11B2HDAC6
SCHEMBL506139 0.70 ESR1 (0.59) ESR1ESR2SMN1; SMN2ABHD6MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120053168-A1 FUSED BENZOAZEPINES AS NEURONAL NICOTINIC ACETYLCHOLINE RECEPTOR LIGANDS TARGACEPT, INC. (US) 2012-03-01 US disclosed
WO-2010096384-A2 FUSED BENZAZEPINES AS NEURONAL NICOTINIC ACETYLCHOLINE RECEPTOR LIGANDS TARGACEPT, INC. (US) 2010-08-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120053168-A1 FUSED BENZOAZEPINES AS NEURONAL NICOTINIC ACETYLCHOLINE RECEPTOR LIGANDS CHRNA2, CHRNA5, CHRNA10 ESR1 1178/4885ESR2 825/4885SMN1; SMN2 395/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.